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1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
(1R,5S,6R)-3-[(2,3,4-trifluorophenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
4-oxo-N-[2-(pyridin-3-yloxy)propyl]-1,4-dihydroquinoline-2-carboxamide
N-[(2-fluorophenyl)methyl]-2-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}acetamide
N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-2-(pyrrolidine-1-carbonyl)piperazine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(pyridin-4-yl)quinoline-4-carboxamide
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
(1R,5R)-6-[(4-methoxy-2,5-dimethylphenyl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(1-benzofuran-2-carbonyl)-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3S,4R)-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
7-(cyclohexylmethyl)-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(4-fluorophenyl)methyl]-4-[1-(2-phenylethyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
7-[(3-methylphenyl)methyl]-2-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
N-ethyl-N-[(1-ethylpyrrolidin-3-yl)methyl]-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
8-fluoro-2-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)quinolin-4-ol
ethyl 3-(2-methoxyethyl)-1-[(2E)-4-methylpent-2-en-1-yl]piperidine-3-carboxylate
N-[(3,4-dimethoxyphenyl)methyl]-N'-(2-fluoro-5-methylphenyl)butanediamide
(3S,4S)-1-(3,5-dimethoxybenzoyl)-4-(3-methoxyphenyl)piperidin-3-ol
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[3-(1H-imidazol-1-yl)propyl]acetamide
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
3-methoxy-1-[4-(4-methylphenoxy)piperidin-1-yl]propan-1-one
(2S,4R)-N-methyl-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]-1-(2-phenylethyl)pyrrolidine-2-carboxamide
1-(furan-2-ylmethyl)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-4-methylbenzamide
N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-3-yl}propanamide
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-5-fluoro-1-methyl-1H-indole
{1-[(1-ethyl-3-methylpiperidin-3-yl)methyl]piperidin-4-yl}methanol
3-[(2R,3R,6R)-5-[3-(methylsulfanyl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(2S,4S)-N-ethyl-1-(furan-3-ylmethyl)-4-[2-(morpholin-4-yl)-2-oxoacetamido]pyrrolidine-2-carboxamide
(4aS,7aR)-1-(5-fluoro-3-methyl-1H-indole-2-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,5-dimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-benzofuran-2-carboxamide
2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-(2-methoxy-5-methylphenyl)acetic acid
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(pyridin-4-ylmethyl)piperidin-2-one
4-(2-cyclopentylacetyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3aR,6aR)-2-(3-methylpyridine-2-carbonyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-(3-chlorophenyl)-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4-diazepane
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,2,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)phenyl]-1H-imidazole
4-(2,4-dioxoimidazolidin-1-yl)-N-[3-(2-ethoxyphenyl)propyl]benzamide
N-[4-(4-{[(1-ethylpiperidin-3-yl)methyl](methyl)amino}piperidin-1-yl)phenyl]-4-methoxybenzamide
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(2-{1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidin-2-yl}ethyl)dimethylamine
[4-(2,1,3-benzoxadiazol-4-ylmethyl)morpholin-3-yl]methanol
2-chloro-4-({1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}methyl)-6-ethoxyphenol
5-cyclopropanecarbonyl-1'-(2,3-dihydro-1H-inden-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1S,5R)-3-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)amine