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(3S,4S)-1-(oxan-4-yl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1-[3-(3-fluorophenyl)benzoyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-(1-methylpiperidin-4-yl)-N-[(1-phenylcyclopentyl)methyl]piperidine-3-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-methylpyrrolidine-3-carboxamide
2-(4-{[(3-hydroxypropyl)(methyl)amino]methyl}phenyl)-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
3-(ethylsulfanyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-(pyridin-4-ylmethyl)propanamide
4-[5-(2,2-dimethylpropanoyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
5-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methyl-3,4-dihydropyrimidin-4-one
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(oxolane-2-carbonyl)-1,4-diazepane
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(methoxymethyl)piperidine
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-6-hydroxypyridine-3-carboxamide
2-(adamantan-1-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)acetamide
methyl 4-(4-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-[1-(1H-imidazol-2-yl)ethyl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,3-oxazole-4-carboxamide
5-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-cyclopentyl-1,4-diazepane
2,2,2-trifluoro-N-{2-[(1-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl)formamido]ethyl}acetamide
2-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-1,3-benzoxazole
3-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-{4-[2-(pyrrolidin-1-yl)ethyl]phenyl}urea
1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-(furan-3-yl)-4-phenyl-1H-imidazole
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[4-ethyl-5-oxo-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
3-[({1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
N-[2-(2-fluorophenyl)-1-[1-(quinolin-5-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3-fluoro-4-methylphenyl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
4-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1-(3-methoxyphenyl)piperazin-2-one
1-methyl-4-({5-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
N-({1-[(3-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-2-(pyridin-4-yl)acetamide
N-benzyl-N-methyl-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-sulfonamide
1-{4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-4-methylpiperazine
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-(oxane-2-carbonyl)piperidine
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[(3-methylpyridin-2-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazine
4-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)phenol
3-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1,2-oxazole-5-carboxamide
1-(4-hydroxy-3-methoxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{1-[(3-methoxyphenyl)methyl]-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl}ethan-1-ol
5-[(1H-indol-4-ylmethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-2-yl)piperazine
3-(2-phenylethyl)-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
propan-2-yl N-{[1-(2,3-dihydro-1H-inden-2-yl)-4-hydroxyazepan-4-yl]methyl}carbamate
4-[(4-fluoro-2-methylphenyl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[(4aR,7aS)-4-(furan-3-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
ethyl 1-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
methyl[2-({5-[(methylsulfanyl)methyl]pyridin-2-yl}oxy)hex-5-en-1-yl](pyridin-3-ylmethyl)amine
(2S,4R)-1-[(2,5-dimethoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)acetamide