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5-chloro-2-{4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine
5-{2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-3-(propan-2-yl)-1,2,4-oxadiazole
4-[(4-fluorophenyl)methyl]-1-(3-fluoropropyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(2S,4R)-4-(dimethylamino)-1-(3-phenyl-1,2-oxazole-5-carbonyl)pyrrolidine-2-carboxylic acid
{4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}methanol
4-(3-chloro-1H-indole-2-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
8-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
(2S)-4-methyl-2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pentanamide
7-(2-methoxyethyl)-2-(2,4,5-trifluorobenzoyl)-2,7-diazaspiro[4.5]decan-6-one
methyl (2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
[(dimethyl-1,2-oxazol-4-yl)methyl][1-(morpholin-4-yl)propan-2-yl]amine
benzyl N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
(1R,5S,6R)-6-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)-3-(2-methylbenzoyl)-3-azabicyclo[3.1.0]hexane
ethyl 1-(4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}benzoyl)piperidine-2-carboxylate
methyl 2-(ethylsulfamoyl)-6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-benzyl-3-butyl-1-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-butyl-N-methyl-3-(morpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-(2-{3-oxo-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-4-yl}ethyl)benzene-1-sulfonamide
4-(2H-1,3-benzodioxol-5-yl)-2-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}phenol
4-{[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzoic acid
N-[(3-methylphenyl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(3-ethoxyphenyl)methyl]-2-ethyl-N-(prop-2-en-1-yl)pyrimidine-5-carboxamide
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-diazepane
1-[(5-chlorothiophen-2-yl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidine
7-(1-methyl-1H-pyrazole-4-carbonyl)-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
5-[(cyclohexylmethyl)amino]-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-acetamido-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]butanamide
8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-(1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
(3aS,6aS)-2-cyclohexyl-5-[(2-methylpyridin-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[5-(cyclopent-3-en-1-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
3-{[4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]methyl}-N-methylbenzamide
2-(3-chloro-4-hydroxyphenyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
4-fluoro-N-({1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}methyl)benzamide
3-cyclopropyl-5-{imidazo[2,1-b][1,3]thiazol-6-yl}-1H-1,2,4-triazole
N-(2-fluorophenyl)-3-{1-[1-(3-methylphenyl)piperidin-4-yl]piperidin-3-yl}propanamide
4-(2,5-dimethylphenyl)-N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)piperazine-1-carboxamide
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2-methoxybenzamide
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-(trifluoromethyl)pyridine
methyl 1-[2-hydroxy-3-(3-{[(3-phenylpropyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
2-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-6-methoxyphenol
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(2-phenoxyethyl)-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2S)-1-hydroxybutan-2-yl]-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-(furan-2-ylmethyl)-9-(2-methoxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
2-(1-tert-butyl-1H-pyrazol-4-yl)-N,8-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine