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methyl (1R,3S,3aR,6aS)-5-methyl-4,6-dioxo-3-(4-phenyl-1,3-thiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]propanamide
N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
1-cyclopentyl-N-(2-hydroxyethyl)-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
3-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-methyl-1-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)urea
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](1H-imidazol-2-ylmethyl)methylamine
2-methyl-5-(propan-2-yl)-N-[2-(1H-1,2,4-triazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-2-(methylsulfanyl)-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-thiazole-4-carboxamide
N-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}acetamide
1-(cyclopropylmethyl)-2-oxo-3-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N,5-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-ethyl-4,6-dimethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(3-fluorophenyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazole
3-phenoxy-N-[1-({[3-(1H-pyrazol-1-yl)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrazine-2-carboxamide
N-[(4-fluorophenyl)methyl]-3-(2-oxopiperidin-1-yl)-N-(pyridin-4-ylmethyl)propanamide
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-propyl-1H-1,2,4-triazole
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-cyclopentylpiperazine
2-methyl-5-{[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrazine
2-methoxy-N-({5-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-methylbenzamide
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
3-cyclopropyl-5-(2,3-dihydro-1H-inden-1-ylmethyl)-1H-1,2,4-triazole
5-fluoro-2-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-1-methyl-1H-indole
5-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
6-chloro-N,N-dimethyl-2-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
ethyl 1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine-2-carboxylate
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-[5-(5-methoxy-3-methyl-1H-indol-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
ethyl 4-{[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]amino}benzoate
3-(2-ethyl-1H-imidazol-1-yl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]propan-1-one
1-{3-[4-(dimethylamino)-5-methylpyrimidin-2-yl]phenyl}ethan-1-one
3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}-1-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3,3,4,4-tetrafluorobutyl)piperidine
2-methyl-4-{5-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]thiophen-2-yl}but-3-yn-2-ol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-({[4-(diethylamino)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-(3-fluoro-4-methoxyphenyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1,2,4-triazin-3-amine
2-[3-(1H-imidazol-1-yl)propyl]-9-(morpholine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R)-2-cyclohexyl-2-hydroxy-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
6-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
6-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
(2S,4R)-4-amino-N-ethyl-1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)pyrrolidine-2-carboxamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-[(3-methylthiophen-2-yl)sulfonyl]piperidine-4-carboxylate
2,4,5-trimethyl-6-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyrimidine
2-ethyl-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]pyrimidine-5-carboxamide
1-ethyl-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-6-oxopiperidine-3-carboxamide
N-{2-[5-(4-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine-4-carboxamide
(2S,4R)-N-ethyl-4-(2-fluorobenzamido)-1-[(3E)-hex-3-enoyl]pyrrolidine-2-carboxamide