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3,3-dimethyl-1-{[5-(naphthalen-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
6-methyl-2-propyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
N3-tert-butyl-1-cyclohexyl-4-oxo-N5-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-one
2-chloro-3-({ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N-(2-methoxyethyl)-4,6-dimethyl-2-oxo-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-[4-(1H-imidazol-2-yl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
2-benzyl-8-(4-methylpiperazine-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2,3-dimethyl-6-[3-(1-methylpiperidin-2-yl)propanoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-2,1,3-benzothiadiazole-4-sulfonamide
[1-(3-methoxyphenyl)ethyl](methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(methoxymethyl)piperidine
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(4-phenylbutanoyl)-decahydro-2,7-naphthyridine-2-carboxamide
2-{1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
1-(3-{[(6-methoxy-2H-chromen-3-yl)methyl]amino}phenyl)pyrrolidin-2-one
methyl 6-[methyl(quinolin-5-ylmethyl)amino]pyrimidine-4-carboxylate
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-4-(1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-2,1,3-benzoxadiazole-5-carboxamide
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-(oxolan-2-ylmethyl)urea
1-{4-[(2-hydroxybutyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-[(2R,3R)-2-hydroxy-1'-(pyridin-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-2-one
(3R)-1-(2,3-difluoro-4-methoxybenzoyl)-3,4,4-trimethylpyrrolidin-3-ol
5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,4-triazole
ethyl 1-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-2-carboxylate
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-(piperidin-1-ylmethyl)benzamide
1-[4-({[1-(2-hydroxyethyl)piperidin-3-yl]methyl}(methyl)amino)piperidin-1-yl]ethan-1-one
[(3R,4R)-1-(1,4-dimethyl-1H-indole-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-methyl-3-{methyl[(5-methylnaphthalen-1-yl)methyl]amino}butanamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-5-oxo-N-(oxolan-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazole-3-carboxamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-4,4,4-trifluorobutanamide
2-(4-methoxy-2-methylphenyl)-2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}acetic acid
N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-6-(propan-2-yl)pyrimidin-4-amine
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
ethyl({[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-ethyl-N-methyl-6-{methyl[(1-phenylpyrrolidin-3-yl)methyl]amino}pyridine-3-carboxamide
N-[2-(5-methylfuran-2-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
1-methyl-4-({4-methyl-5-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
6-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-sulfonyl]-1,2,3,4-tetrahydroquinolin-2-one
7-(furan-2-carbonyl)-2-methyl-N-[(2R)-oxolan-2-ylmethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2-{[(3R,5S)-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidin-3-yl]formamido}ethyl)acetamide
N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-methoxybenzamide
N-({5-[(trimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(cyclopropylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(hydroxymethyl)-4-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-methylpyridin-3-ol
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)furan-2-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(4-fluoro-2-methylbenzoyl)pyrrolidin-3-yl]methanol
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(5-fluoro-2-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid