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2-{1-[(2-methylphenyl)methyl]-4-(quinolin-8-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(piperidine-1-carbonyl)benzene-1-sulfonamide
4-[(4-fluorophenyl)methyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-(pyridin-2-ylmethyl)piperidin-4-amine
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-2-ol
N-cyclopropyl-3-{[1-(3,5-difluorophenyl)ethyl]sulfamoyl}benzamide
1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N3-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}piperidine-1,3-dicarboxamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[2-(pyrazin-2-yl)ethyl]propanamide
4-[(3,4-difluorophenyl)methyl]-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]phenol
2,3-dimethoxy-N-{[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]methyl}benzamide
(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
1-(3-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenyl)ethan-1-one
1-(3-hydroxyadamantan-1-yl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
2-{5-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]furan-2-yl}-1-methyl-1H-1,3-benzodiazole
N-(1-cyclopropylethyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
4-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-4-oxobutanamide
1-tert-butyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-oxopyrrolidine-3-carboxamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
(2-methoxyethyl)({4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}methyl)amine
4-(2-hydroxy-4-methylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
(2R,3R,6R)-5-[3-(1H-imidazol-1-yl)propyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[2-methyl-4-(4-methylphenyl)-5-oxopiperazine-1-carbonyl]benzonitrile
N-ethyl-4-hydroxy-2-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
6-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-2-carbonitrile
4-[(dimethylamino)methyl]-1-[3-(1H-pyrazol-1-yl)benzoyl]azepan-4-ol
[(4-{[1-(furan-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
1-(6-fluoro-4-methylquinolin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-3-yl]methanol
2-{[(2,3-difluoro-4-methoxyphenyl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
5-acetyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-2-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
N-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
N,1-dimethyl-N-(2-phenylethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3aS,6aS)-2-[(3,4-difluorophenyl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[(2-ethylphenyl)carbamoyl]phenyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
N-{2-[(1-methoxypropan-2-yl)amino]ethyl}-3-methylpyridin-4-amine
1-(cyclopropylmethyl)-N-ethyl-5-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-[3-(piperidin-1-ylmethyl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)-1-[(2-methoxyphenyl)methyl]piperidine
2-[(1-ethylpyrrolidin-2-yl)methyl]-6-(morpholine-4-carbonyl)-2,3-dihydro-1H-isoindol-1-one
6-(2-methylphenyl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]pyrrolidine-2-carboxamide
1-[(4aR,8aR)-4a-hydroxy-7-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
4-hydroxy-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2-(6-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-methylpyrimidin-4-yl)ethan-1-amine
N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide