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2-[4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methoxy)phenyl]acetamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-(thiophen-2-ylmethyl)pyrimidin-2-amine
4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-methyl-3,4-dihydro-2H-1,4-benzothiazin-3-one
methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
5-methyl-1'-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[2-(2,4-difluorophenoxy)propanoyl]-1-(2-methylphenyl)piperazin-2-one
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-(pyridin-4-yl)propanamide
N-ethyl-4-[(1-phenoxypropan-2-yl)amino]piperidine-1-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)ethan-1-one
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one
2-[5-(2-fluoro-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]-N-methylethane-1-sulfonamide
(benzylsulfamoyl)[2-methoxy-1-(pyridin-2-yl)ethyl]amine
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
3-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-(3-methoxyphenyl)-3-[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]propanamide
8-(2,6-dimethylpyrimidine-4-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(2,5-dimethylbenzoyl)-2-(3-phenylpropyl)morpholine
2-(4-fluorophenyl)-N-(1,2-oxazol-3-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
9-[(2-ethylpyrimidin-5-yl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
ethyl 2-[2-(1H-imidazol-1-ylmethyl)pyrrolidin-1-yl]-6-methylpyrimidine-4-carboxylate
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
N-[(3-methoxyphenyl)methyl]-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-3-yl}propanamide
3-ethoxy-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]propanamide
[1-(4-methoxybenzenesulfonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2-(oxolane-2-carbonyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2,2-dimethyl-5-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]thiomorpholin-3-one
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-N-(4-methoxyphenyl)acetamide
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
N,N,7-trimethyl-3-{[(2-methylpropyl)amino]methyl}quinolin-2-amine
7-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroquinoxalin-2-one
2-(1-{[1-(1,4-dithiepan-6-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-methyl-1,4-diazepane
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-4-(piperazine-1-carbonyl)benzene-1-sulfonamide
N-(1-{1-[(4-fluorophenyl)methyl]-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl}butyl)acetamide
(3S,9aR)-8-[(3,4-dimethylphenyl)methyl]-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3aS,7aR)-2-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-({2-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)-4-methylpiperidine-4-carbonitrile
5-cyclopropyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,3,4-oxadiazol-2-amine
4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-[4-(benzyloxy)-3-fluorophenyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
N-[(1-cyclohexyl-1H-1,2,4-triazol-5-yl)methyl]methanesulfonamide
1-[(2S)-2,3-dihydroxypropyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-6-(cyclobutylmethyl)-3-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-ethyl-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-1,2,3-thiadiazole-5-carboxamide
2-[3-oxo-9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-2-(trifluoromethyl)morpholine
N-{1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}pyrimidin-2-amine
N-{[1-(2,2-dimethylpropyl)piperidin-3-yl]methyl}-5-methylpyridine-3-carboxamide