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2-(dimethyl-1,3-thiazol-5-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]propan-1-one
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[3-(methylamino)propyl]propanamide
4,6-dimethyl-1-{3-oxo-3-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propyl}-1,2-dihydropyrimidin-2-one
6-(2-fluorophenyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
7-[(3,4-difluorophenyl)methyl]-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
1-(4-ethylpiperazin-1-yl)-3-(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-yl)propan-1-one
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]propan-1-one
2-(3-fluoro-4-methylphenyl)-2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}acetic acid
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1,3-benzothiazole-5-carboxamide
1-(2-methyl-1,3-thiazole-5-carbonyl)-3-(4-methylphenoxymethyl)piperidine
ethyl 1-[3-(methoxycarbonyl)benzoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
N-[(3R,4S)-4-cyclopropyl-1-(4-methylpent-3-en-1-yl)pyrrolidin-3-yl]-1-(1H-imidazol-1-ylmethyl)cyclopropane-1-carboxamide
[(3S,7S)-5-(2,4-dimethoxybenzoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
5-{1-[2-(4-methoxyphenoxy)ethyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
3-methyl-N-(oxolan-2-ylmethyl)-1-propyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
6-(4-methyl-1H-pyrazol-1-yl)-1H-indole
2-(2-methyl-1,4-oxazepane-4-carbonyl)-3,4-dihydroquinazolin-4-one
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
1-{2-oxo-2-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
4-[(3-methylphenyl)sulfanyl]-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
(2E)-1-[7-(6,7-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(thiophen-2-yl)prop-2-en-1-one
3-({[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amino}methyl)-N-(pyrazin-2-yl)benzamide
2-ethyl-4-methyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,3-oxazole-5-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
dimethyl({4-methyl-5-[1-(4-methylpiperazine-1-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
(1S,5R)-3-cyclobutanecarbonyl-6-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]-1,3-thiazole-4-carboxamide
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
5-({ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-N,N-dimethylpyridin-2-amine
N-[(5-{[4-(difluoromethoxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-[(2-fluorophenyl)methyl]piperazin-2-one
(3S,4R)-1-[(5-ethylpyridin-2-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(3aR,6aR)-2-methanesulfonyl-5-{2-methylthieno[2,3-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-methoxy-4-(prop-2-en-1-yl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
9-(4,6-dimethylpyrimidin-2-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetyl)-1,4-diazepane-1-carbaldehyde
1-(3-chloropyridin-2-yl)-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
(2S,4R)-4-{[(2,4-difluorophenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-ethyl-N-methyl-4-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-sulfonamide
2-(3-acetyl-1H-indol-1-yl)-1-(4-methyl-1,4-diazepan-1-yl)butan-1-one
ethyl 3-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)formamido]propanoate
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-[(2-cyclohexylpyrimidin-5-yl)methyl]-N-methylthian-4-amine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5,6-dimethylpyrimidin-4-amine
N-methyl-N-(1-{1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-2-phenylethyl)thiophene-2-carboxamide
2-[1-(3-fluorophenyl)-5-[1-(2-methoxyacetyl)piperidin-3-yl]-1H-1,2,4-triazol-3-yl]acetamide
4-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1,2,5-oxadiazole-3-carboxamide