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(3S,4S)-1-[1-(3,5-dimethylphenyl)piperidin-4-yl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-[3-(cyclopentyloxy)propyl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N'-[2-(propan-2-yl)phenyl]butanediamide
4-[5-benzoyl-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
4-methoxy-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)cyclohexane-1-carboxamide
5-chloro-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(methylsulfanyl)acetamide
1-{4-[hydroxy(pyridin-3-yl)methyl]piperidin-1-yl}-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-ethyl-4-phenyl-9-(pyridazine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1,4-dithiepan-6-amine
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-3-(4H-1,2,4-triazol-4-yl)propanamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-1-methylcyclopropane-1-carboxamide
N-[4-(4-{[(1S)-1-carbamoyl-2-phenylethyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
(5S,9aS,9bS)-5-(2,3-dimethoxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-(4-phenylpiperazin-1-yl)-5-[2-(1H-pyrazol-4-yl)ethyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
9-methoxy-7-oxo-3-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(6-hydroxypyrimidin-4-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}oxolane-2-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
5-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
2-(2-methoxy-4-methylphenoxymethyl)-4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1,3-oxazole
3-[5-(1-phenylcyclohexanecarbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
(1S,5R)-3-(pyrimidin-2-yl)-6-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N,2-dimethyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)(quinolin-8-ylmethyl)amine
[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
methyl 3-(4-{[4-(3-fluorophenoxy)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
2-[2-(methylsulfanyl)pyrimidin-4-yl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-[2-(benzylsulfanyl)-4-hydroxypyrimidine-5-carbonyl]-1,4-oxazepan-6-ol
2-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1,2-dihydrophthalazin-1-one
6-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}pyridine-2-carboxylic acid
3-(4-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenyl)prop-2-yn-1-ol
4-amino-2-({[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}amino)pyrimidine-5-carbonitrile
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}thiophene-3-carboxamide
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2-hydroxybenzoic acid
5-{[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]sulfonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-6-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-(ethylamino)-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]pyrimidine-5-carboxamide
3-butyl-4-(2-chlorobenzenesulfonyl)-1-methylpiperazin-2-one
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
5-cyclopentyl-3-{[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,2,4-oxadiazole
3-[4-(3,4-difluorobenzoyl)piperidine-1-carbonyl]piperidine-1-carboxamide
5-ethyl-N-[4-(oxolan-2-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-(2-methylpropyl)-1-(2-phenylethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-cyclopropyl-5-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1H-1,2,4-triazole
5-benzyl-3-methyl-5-(piperidin-4-yl)imidazolidine-2,4-dione