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3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-N-(3-methylphenyl)piperidine-1-carboxamide
2-[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carbonyl]pyridine
(2R,3R)-1'-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-N-(2,3-dihydro-1H-inden-5-yl)-5-(methylsulfamoyl)benzamide
N-({4-[(dimethylamino)methyl]phenyl}methyl)cyclohex-3-ene-1-carboxamide
3-(3-amino-4-fluoro-1H-indazol-1-yl)-5-(azepane-1-sulfonyl)benzoic acid
2-(1-benzyl-1H-pyrazol-4-yl)-N-ethyl-N-methylquinoline-4-carboxamide
[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(thiophen-2-yl)-1H-pyrazol-4-yl]methanol
N-[(6-chloropyridin-3-yl)methyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
ethyl 4-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
3-{5-cyclopentyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3,5-dimethylphenyl)-1H-pyrazole
3-[(3-fluorophenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(2-methoxyphenoxy)-N-[(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
2-(2-amino-4-methyl-1,3-thiazol-5-yl)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
1-cyclopropyl-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1H-pyrrole-2-carboxamide
N,3,6-trimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-benzofuran-2-carboxamide
[(2S,6S)-4-cycloheptanecarbonyl-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
bis(1,3-oxazol-4-ylmethyl)({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-amino-1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
3-{[1-(2,6-dimethoxypyrimidine-4-carbonyl)piperidin-4-yl]methyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 4-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]piperidine-1-carboxylate
2-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
5-({3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}methyl)-2,1,3-benzoxadiazole
N-[(1-methylpiperidin-4-yl)methyl]-2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]acetamide
3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1-[3-(1H-pyrazol-1-yl)phenyl]urea
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-1,2,3-thiadiazole-4-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
N-{2-[methyl(2-phenylethyl)amino]ethyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
3-[4-(4-ethoxy-3-methylphenyl)-4-oxobutanamido]-4,4,4-trifluorobutanoic acid
1-(4,7-dimethylquinazolin-2-yl)-N-(thiophen-2-ylmethyl)azepan-4-amine
1-ethyl-3-{4-phenyl-1-[(3-propyl-1,2-oxazol-5-yl)methyl]-1H-imidazol-5-yl}piperidine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-(6-methyl-2H-1,3-benzodioxol-5-yl)urea
3-methyl-1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]but-2-en-1-one
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3,4-dihydroquinazolin-4-one
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl][(1-ethylpyrrolidin-2-yl)methyl]{[1-(2-methoxyethyl)piperidin-4-yl]methyl}amine
3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-N-methylpyridin-2-amine
7-methoxy-N-[(5-methoxy-1H-indol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-(3-fluoro-2-methylphenyl)-2-[(morpholin-2-ylmethyl)amino]acetamide
N,N-dimethyl-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(trifluoromethyl)pyrimidin-4-amine
1-benzyl-N3-ethyl-N5-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-methyl-6-(pyridin-4-yl)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-4-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,2-dihydrophthalazin-1-one
2-methyl-5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
N-[(1R,3R)-3-aminocyclopentyl]-6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide