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3-({[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)pyridin-2-amine
1,3-dimethyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-hydroxy-5-{[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}benzoic acid
3-{[1-(3-hydroxypyridine-2-carbonyl)pyrrolidin-3-yl]methyl}benzamide
1-[4-(morpholin-4-ylmethyl)phenyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
1-benzyl-N3-[2-(4-chlorophenyl)ethyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[(5-methylthiophen-2-yl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
9-[(2-ethoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-chlorophenyl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(prop-2-en-1-yl)acetamide
ethyl 4-[(1-{4-[2-(4-methoxyphenyl)acetamido]phenyl}piperidin-4-yl)amino]piperidine-1-carboxylate
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3-fluoro-2,4-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{1-[4-(2,5-dimethoxybenzoyl)benzoyl]piperidin-3-yl}pyrimidine
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(3-methoxyphenoxymethyl)piperidine
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(pyridin-2-ylmethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-{5-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}phenol
4-methoxy-2-{[4-(4,6,7-trimethylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}phenol
1-(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)-4-(2-methoxyethyl)piperazine
3-methyl-6-(3,4,5-trifluorophenyl)pyridazine
6-methyl-4-(4-oxo-4H-chromen-3-yl)-7-(2-oxopyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
7-(4-chlorophenyl)-2-(furan-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[2-(2-fluorophenyl)ethyl]-3-[(4-hydroxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-2-(2-phenylethyl)-1,3-benzoxazole
1-cyclopropyl-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-1H-pyrrole-2-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(2-methylbutanoyl)piperidin-4-yl]oxy}benzamide
3-methanesulfonyl-N-[(3R,4S)-1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]propanamide
1-[1-(5-methyl-1H-indazole-3-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
3-[(4aR,8aR)-octahydro-2H-1,4-benzoxazine-4-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N-[(2-{3-[2-(4-methoxyphenyl)acetamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-4-methyl-1H-imidazole-2-carboxamide
2-{2-[3-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}acetamide
4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyrimidin-2-amine
N-(2-{4-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]phenoxy}ethyl)acetamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(3,4-dichlorophenyl)-4-(pyridin-2-ylmethyl)morpholine
1-[2-hydroxy-3-(4-methoxy-2-{[methyl(oxan-4-ylmethyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-fluoro-1H-indole
N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}propanamide
3-{1-[4-phenyl-5-(1,3-thiazol-2-yl)-1H-imidazol-1-yl]propyl}pyridine
1-{3-[2-(4-methyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]phenyl}imidazolidin-2-one
N-cyclobutyl-3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]acetamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
1-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
1-(3-methylpyridin-2-yl)-4-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperazine
2-[4-(2-methyl-4-phenylpyrimidine-5-carbonyl)morpholin-3-yl]-1-(pyrrolidin-1-yl)ethan-1-one
4-{4-[3-(2-fluorophenoxy)azetidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}pyridine
2-(2-ethoxypyridin-3-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one