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(5-{1-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
{3-[(4-fluorophenyl)methyl]-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl}methanol
2-(4-ethylpiperazin-1-yl)-N-(3-hydroxy-2,2-dimethylpropyl)-2,3-dihydro-1H-indene-2-carboxamide
ethyl 1-[3-(methylsulfanyl)propanoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
1-(1,3-thiazol-2-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
3-butyl-4-{2-[4-(hydroxymethyl)phenyl]acetyl}-1-methylpiperazin-2-one
6-methyl-5-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,N-dimethyl-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine-1-carboxamide
3-[3-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methoxy-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
(2S,3R)-2-amino-3-hydroxy-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}butanamide
4-[1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperidin-4-yl]pyrimidine
2-(1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidin-2-yl)pyridine
N-methyl-N-(1H-pyrazol-3-ylmethyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
[5-methyl-7-(quinolin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
1-(2H-1,3-benzodioxol-5-ylmethyl)-N-(1H-imidazol-2-ylmethyl)-6-methyl-4-oxo-2-propyl-1,4-dihydropyridine-3-carboxamide
2,3-dimethyl-7-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
4-ethyl-3-({1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-2-(2-oxopiperidin-1-yl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
2-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-4-methylphenol
1-(4-hydroxypiperidin-1-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-5-{4-[1-(propan-2-yl)piperidine-3-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1,6-dimethyl-3-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
8-fluoro-3-(quinolin-6-ylmethyl)-3,4-dihydroquinazolin-4-one
5-chloro-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}pyridine-2-carboxamide
1-(3-{[(2,2-dimethylpropyl)(methyl)amino]methyl}phenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
N-{2-[(1-acetylpiperidin-3-yl)formamido]ethyl}-4-fluorobenzamide
N-[(4-methoxypyridin-2-yl)methyl]-N-methyl-2-oxo-1-phenylpyrrolidine-3-carboxamide
2-(methoxymethyl)-N-[3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
4-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-yl}benzoic acid
1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
7-methyl-2-(1-methyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
9-[3-(methylsulfanyl)propyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(3-fluorophenoxy)piperidin-1-yl]propan-1-one
(1S,4S)-2-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
4-(4-ethoxy-3-methylphenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-oxobutanamide
N-cyclopropyl-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetamide
1-methanesulfonyl-4-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1,4-diazepane
2-chloro-N-ethyl-4-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)benzamide
1-(oxolan-3-ylmethyl)-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
1-[2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butanoyl]-1,4-diazepan-5-one
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(ethyl)(2-methoxyethyl)amine
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
(3S)-3-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}azepan-2-one
8-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one