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6-(oxolan-3-yl)-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
methyl[2-(morpholin-4-yl)ethyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
2-(4-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
2-[5-(2,3-difluorophenyl)-1H-indazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
2-({4-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
5-{2-[(4aS,7aR)-4-(2-methoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]ethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-methoxy-N-{[1-(3-methoxypropanoyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
1-[2-(thiophen-2-yl)-1,3-thiazole-4-amido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
1-{3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-(2-methoxyphenyl)-3-[(thian-4-yl)amino]propanamide
3-[({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)methyl]-1λ6-thiolane-1,1-dione
8-[(3-chloro-4-fluorophenyl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-[(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}pyrimidin-4-yl)(methyl)amino]propane-1,2-diol
2-methyl-5-({3-[4-(5-methylfuran-2-yl)-1H-1,2,3-triazol-1-yl]propyl}sulfanyl)-1,3,4-thiadiazole
N-(2-methoxyethyl)-3-(1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
4-methyl-2-{2-oxo-2-[4-(2-oxo-1,3-oxazolidin-3-yl)piperidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
2-[(4-chlorophenyl)methyl]-N-[(5-methylpyrazin-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
(2R,6S)-4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-2,6-dimethylmorpholine
4-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
2-cyclopropyl-8-[4-(4-fluorophenyl)-4-oxobutyl]-2,8-diazaspiro[5.5]undecan-3-one
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)(thiophen-2-ylmethyl)amine
4-(1H-pyrazol-3-yl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidine
4-oxo-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
5-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}-2-(furan-2-yl)pyrimidine
1-ethyl-2-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
4-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]benzoic acid
3-ethyl-N,4-dimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-({2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(propan-2-yl)-9-(quinolin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-4-methylpiperidine-3,4-diol
N-ethyl-3-(2-methoxyphenyl)-N-[2-(3-methylphenoxy)ethyl]-1H-pyrazole-5-carboxamide
2-{2-[(2-methyl-1,4-oxazepan-4-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-(2-hydroxyethyl)-3-(1H-imidazol-2-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
1-(2-ethoxyethyl)-2-oxo-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(2,2,2-trifluoroethyl)piperazine
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
(3aR,5S,6S,7aS)-2-[4-(1H-pyrazol-3-yl)benzoyl]-octahydro-1H-isoindole-5,6-diol
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
2-methoxy-6-{[3-(pyridine-2-carbonyl)piperidin-1-yl]methyl}phenol
3-(piperidin-3-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
8-(4-chloro-2-methoxybenzoyl)-1-oxa-8-azaspiro[4.5]decane
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N5-[(5-chlorothiophen-2-yl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3,5-dichloro-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,4-dimethylbenzamide
4-(4-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}phenyl)morpholine