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5-({2-[(4-methoxyphenyl)methyl]morpholin-4-yl}methyl)-2,1,3-benzoxadiazole
1-methyl-1-(1-methylpiperidin-4-yl)-3-(5-pentyl-1,3,4-thiadiazol-2-yl)urea
N-(4-fluorophenyl)-1-(3-methylfuran-2-carbonyl)piperazine-2-carboxamide
N-[(3S,4R)-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(1-{1-[3-(4-fluorophenyl)phenyl]piperidin-4-yl}piperidin-3-yl)methanol
3-{1-[(2,3-difluorophenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
(3S,4S)-1-[(4-methoxypiperidin-1-yl)sulfonyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-(6-methyl-2-phenyl-1,2-diazinane-1-carbonyl)-2-(thiophen-2-yl)pyrimidin-4-ol
4-(5-chloro-2-methoxybenzoyl)-1-phenylpiperazin-2-one
2-[2-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
4-benzyl-3-ethyl-1-(2-hydroxy-3-methoxybenzoyl)-1,4-diazepan-5-one
[1-(5-chloro-2-methylpyrimidine-4-carbonyl)-3-(cyclopropylmethyl)piperidin-3-yl]methanol
1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-(4-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]sulfonyl}phenyl)-3-methylurea
2-[(3-methylquinoxalin-2-yl)methyl]-2-azaspiro[4.4]nonan-3-one
2-[4-(ethylamino)pyrimidin-2-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
dimethyl(3-{2-[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
(3R,4R)-1-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]-4-cyclobutyl-3-methylpiperidin-4-ol
2-(5-methyl-1H-pyrazol-1-yl)-1-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}ethan-1-one
(3S,4S)-4-(4-fluorophenyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-ol
1-{5-[(2,6-difluorophenyl)methyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine
4-ethyl-5-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
8-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-(2-fluoro-5-methylphenyl)-N'-[(1R)-1-(4-fluorophenyl)ethyl]butanediamide
5-(morpholin-4-yl)-2-(pyrrolidin-3-ylmethyl)-2,3-dihydropyridazin-3-one
3-{1-[3-(3-hydroxy-3-methylbutyl)phenyl]-N-methylformamido}-N-methylbutanamide
4-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-1-oxaspiro[4.5]decan-2-one
4-(4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
5-acetyl-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methylthiophene-2-carboxamide
3-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-2,2-dimethylpropan-1-ol
(2S,4R)-N-methyl-1-(oxan-4-yl)-4-[2-(thiophen-2-yl)acetamido]pyrrolidine-2-carboxamide
3-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]-1,6-dimethyl-1,4-dihydroquinolin-4-one
2-[2-(azepan-1-ylmethyl)phenyl]-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
N-[(3R,4R)-3-hydroxy-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl]pyridine-2-carboxamide
N-{2-benzyl-1-methyl-7-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}propanamide
2-[(1-benzyl-1H-indol-3-yl)sulfanyl]-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
4-hydroxy-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
N,N-dimethyl-2-[(3-{[(3-methyl-1,2-oxazol-5-yl)methyl]sulfamoyl}phenyl)formamido]acetamide
1-(2-chlorophenyl)-4-[2-(2-chlorophenyl)-2-hydroxyacetyl]piperazin-2-one
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
1-(4-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl](methyl)amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
(3aR,6aR)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyridine-4-carboxamide
N-[1-(pyrimidin-2-yl)piperidin-4-yl]-1-azabicyclo[2.2.2]octan-3-amine
1-methanesulfonyl-4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperazine
(3S,9aR)-3-[(2S)-butan-2-yl]-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione