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N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
4-({2-[(cyclobutylformamido)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)benzoic acid
methyl (1R,3S,3aR,6aS)-5-methyl-4,6-dioxo-3-(6-phenoxypyridin-3-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-benzoxepine-4-carboxamide
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,3,4-trimethyl-5-sulfamoylbenzamide
N-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methylcyclohexanamine
4-(1-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)-2,1,3-benzoxadiazole
6-ethyl-2-methoxy-3-{[(2-methyl-5-propylpyrimidin-4-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
8-fluoro-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}quinoline
4-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(4-methylpyridin-2-yl)propyl]benzamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
6-[1-(4-chloro-3-methylbenzoyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
1-methyl-N-[(5-methylfuran-2-yl)methyl]-5-[(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-fluoro-N,2-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]quinoline-4-carboxamide
1-{[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]methyl}pyrrolidin-2-one
1-methyl-N-{3-[methyl(phenyl)amino]propyl}azepane-2-carboxamide
(1R,5R)-3-(4-methylpyridine-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-propyl-1,3-thiazole
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[3-(pyrazin-2-yl)propanoyl]piperidine-3-carboxylate
2-(2-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-4-(pyridin-3-yl)phenoxy)acetic acid
N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydronaphthalen-1-amine
N-methyl-6-(propane-2-sulfonyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
5-(2-methoxypyridin-3-yl)-3-(4-phenylpiperazin-1-yl)pyrazin-2-amine
3-(1H-1,3-benzodiazol-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}propanamide
N-(3,4-dimethoxyphenyl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-amine
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-cyclobutyl-6-methylpyrimidin-2-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-[(prop-2-en-1-yl)amino]benzamide
pyridin-2-yl(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)methanol
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
5-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}-2,1,3-benzothiadiazole
2-(3-methylphenyl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]acetamide
N-(2-methoxy-5-methylphenyl)-2-{[1-(propan-2-yl)piperidin-4-yl]formamido}acetamide
(1S,5R)-3-(4-chloro-2-methoxybenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
[(2S,6S)-4-[(5-ethylfuran-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-methyl-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
methyl 2-[(3-fluorophenyl)sulfamoyl]-6-(4-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{3-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}pyrrolidin-2-one
[(3R,4R)-1-[(2-fluoro-5-methylphenyl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
5-[2-(2-methoxyethyl)piperidine-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
4-(2,5-dimethylthiophen-3-yl)-2-[5-methyl-4-(2-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-(3-hydroxy-3-phenylpropyl)-N-methylpropanamide
4-(1H-1,3-benzodiazol-1-yl)-1-methylpiperidine-4-carboxylic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(diethylamino)-3-[5-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
5,5-dimethyl-1-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione