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1-[3-({methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amino}methyl)phenyl]ethan-1-one
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazole
1-[2-(dimethylamino)ethyl]-5-oxo-N-[(2,4,5-trifluorophenyl)methyl]pyrrolidine-3-carboxamide
N-[2-(1-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}piperidin-2-yl)ethyl]acetamide
N-{[(2S,4S)-4-fluoro-1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl]methyl}pyrrolidine-1-carboxamide
(4aR,7aS)-1-ethyl-4-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(5-chlorofuran-2-yl)methyl]-2-(2-methoxyethyl)morpholine
1-ethyl-N,N-dimethyl-3-[2-(methylsulfanyl)phenyl]-1H-1,2,4-triazol-5-amine
2-methyl-9-[2-(methylamino)acetyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-{[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}benzonitrile
2-methoxy-3-{[(oxan-4-yl)amino]methyl}-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-(1-cyclopentyl-1H-pyrazol-5-yl)-4-(3-methylphenyl)piperazine-1-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(4-methylpyridin-2-yl)propyl]acetamide
2-[1-(3-methylbutyl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-4-methylpentane-1,2-dione
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-benzyl-4-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]morpholine
5-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
2-{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(3,4-difluorophenyl)methyl]piperidine-4-carboxamide
5-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-{[3-(azepane-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl](methyl)amino}ethan-1-ol
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]benzamide
(2H-1,3-benzodioxol-4-ylmethyl)({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[2-(methylsulfanyl)ethyl]amine
4-(2-aminopyridine-4-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-[1-(3,4-dimethylphenyl)-5-[2-(N-methylmethanesulfonamido)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-amine
1-(5-methoxy-2-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
9-(6-cyclopropylpyrimidin-4-yl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}({[4-(pyrimidin-2-yloxy)phenyl]methyl})amine
5-hydroxy-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]pyrazine-2-carboxamide
6-methyl-5-[5-(4-propylpyrimidin-5-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[1-(pyridin-3-yl)propan-2-yl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
3-[(carbamoylmethyl)sulfamoyl]-N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]benzamide
4-(1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidin-4-yl)morpholine
2-[(6-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}pyrimidin-4-yl)amino]ethan-1-ol
2-[2-(furan-2-yl)phenyl]-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-imidazole
2-(2,3-dihydro-1H-isoindol-2-ylmethyl)quinolin-4-ol
(1S,6R)-9-(5-propylthiophene-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{6-hydroxy-4-[2-(1H-imidazol-4-yl)acetyl]-1,4-diazepan-1-yl}pyridine-3-carbonitrile
2-({4-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
2-butyl-4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide