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3-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-4H-chromen-4-one
N-methyl-2-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-N-(propan-2-yl)acetamide
(1R,5S)-3-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
benzyl({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
2-methyl-6-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)pyrimidin-4-ol
(2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
2-[4-(2-phenoxyethyl)phenyl]acetamide
5-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-3-yl]-N-[(2-methoxyphenyl)methyl]-4-methyl-1,3-thiazol-2-amine
3-(4-methyl-1,3-thiazol-5-yl)-1-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}propan-1-one
1-({2,5-dimethyl-3-[(2-methylpiperidin-1-yl)methyl]phenyl}methyl)-1,4-diazepan-5-one
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(4-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}piperazin-1-yl)pyridine-3-carbonitrile
[(3,4-dichlorophenyl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
3,5-dimethyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-benzofuran-2-carboxamide
2-methyl-6-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,3-benzothiazole
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-(propan-2-yl)oxane-4-carboxamide
(3aR,6aR)-2-cyclopentanecarbonyl-5-(3-fluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-butyl-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
4-chloro-2-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenol
6-[4-(4-methoxyphenyl)butan-2-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]acetamide
5-methoxy-1-methyl-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
1-ethyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-[(1R,5S)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4-hydroxyphenyl)propan-1-one
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(3-fluorophenyl)methyl]piperidin-3-yl}propanamide
5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-2,1,3-benzoxadiazole
5-fluoro-2-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
5-{5-[(3-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}quinoline
1-(1,3-oxazole-5-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
4-(1-{2-[(dimethylcarbamoyl)amino]acetyl}piperidin-3-yl)benzoic acid
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1-(pyrimidin-2-yl)piperidine-4-carboxamide
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2-(pyridin-2-ylsulfanyl)acetamide
N-(1-methoxypropan-2-yl)-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazol-3-yl]-4-methyl-N-[(2,3,4-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
{1-[3-(thiophen-3-yl)propyl]piperidin-4-yl}methanol
1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
2-{[(3S,4R)-4-methoxyoxolan-3-yl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(3S,4R)-1-[1-(2-chlorobenzoyl)piperidine-4-carbonyl]-4-methylpiperidine-3,4-diol
N-[(5-chlorothiophen-2-yl)methyl]-2-(morpholin-2-yl)acetamide
1-(2-propyl-1,3-thiazole-4-carbonyl)-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
1-methyl-2-oxo-8-[2-(1H-pyrazol-1-yl)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(dimethylamino)-8-[(8-methoxyquinolin-2-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)piperazine-1-carboxamide
N-benzyl-5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-(5-acetylthiophen-3-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[(3-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-1,4-dioxane-2-carboxamide
1-{2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
methyl 4-({[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)benzoate