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N-{4-oxo-4-[3-oxo-4-(2-phenylphenyl)piperazin-1-yl]butyl}acetamide
2-(methylsulfanyl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
(2S)-N-(1H-indazol-4-yl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-2-(pyrrolidin-1-yl)propanamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethyl-1,3-oxazole-4-carboxamide
3-(methylsulfanyl)-N-[(1S,2R)-2-{[1-(pyrazine-2-carbonyl)piperidin-4-yl]amino}cyclobutyl]propanamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
3-[1-(3-phenoxypropanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
5-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-4-phenylpyrimidin-2-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-4-(piperidin-3-yl)benzamide
N-[(2,4-difluorophenyl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(2,5-difluorophenyl)ethan-1-one
2-(1H-imidazol-1-yl)-1-[4-(thiomorpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
(4aR,7aS)-1-methyl-4-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(thiophen-2-ylmethyl)butanamide
N-(2,3-dihydro-1H-inden-2-yl)-1-[4-(1H-pyrazol-5-yl)phenyl]piperidin-4-amine
3-{[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-(propan-2-yl)-1,2,4-oxadiazole
4-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}butan-1-ol
6-{[(2,6-difluorophenyl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-methyl-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
7-[(5-methylthiophen-2-yl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(9aR)-8-[(3-fluorophenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aR,8aS)-1-(cyclohexylmethyl)-6-[(2-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
3-ethyl-5-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1,2-oxazole-4-carboxamide
5-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
3-(2,4-dimethoxybenzoyl)piperidine
3-cyclohexyl-5-{[2-(pyrrolidin-1-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-1,2-oxazole
(2R,6R)-4-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-{1-[2-(dimethylamino)benzoyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
1-cyclopentyl-4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{4-[1-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]phenyl}-1H-1,2,4-triazole
2-(1H-indol-3-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
6-cyclopentyl-1-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-[(4-methanesulfonylphenyl)methyl]-3-methyl-3,9-diazaspiro[5.6]dodecane
6-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl 5-[2-(3,4-dimethylphenoxy)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
(1S,5R)-6-benzyl-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(3-methoxypropyl)-3-(4-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
7-(1,3-benzothiazol-2-yl)-4-(2,2-dimethylcyclopropanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(1S,2R)-2-aminocyclobutyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(3R,4R)-1-[(2-methoxyquinolin-3-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-4-methyl-N-(pyridin-4-ylmethyl)benzamide
N,N-diethyl-1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}pyrrolidin-3-amine
5-[5-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]thiophene-2-carboxylic acid
[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]diphenylmethanol
2-amino-4-methyl-N-(pentan-3-yl)-N-(2-phenylethyl)pyrimidine-5-carboxamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-(naphthalen-2-yloxy)propanamide
2-(1-benzyl-4-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
1-(4-{[(1-ethylcyclobutyl)methyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one