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(2S,4S)-4-amino-1-({1-[(2-fluorophenyl)methyl]-1H-indol-3-yl}methyl)-N-methylpyrrolidine-2-carboxamide
2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}benzene-1,3-diol
2-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
ethyl 1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
methyl (2S)-2-({[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]carbamoyl}amino)propanoate
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}piperazine
8-(2-aminopyrimidin-4-yl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(2-fluorophenyl)methyl]-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)propanamide
2-phenyl-4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}morpholine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)(2-methylpropyl)(pyridin-2-ylmethyl)amine
2-(1,4-dimethylpiperazin-2-yl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(methoxymethyl)-1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)pyrrolidine
N-methyl-4-oxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(3S,4R)-4-(pyridin-3-yl)-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}pyrrolidine-3-carboxylic acid
2-[3-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenoxy]ethan-1-ol
6-methoxy-3-methyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]-1-benzofuran-2-carboxamide
6-methyl-3-[3-(1H-pyrazol-1-yl)phenyl]pyridin-2-amine
2-({4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
N-(5-oxo-1-propylpyrrolidin-3-yl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-5-methanesulfonyl-N,2-dimethylpyrimidin-4-amine
1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
(4S)-3,3,4-trimethyl-1-({2-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperidin-4-ol
5-acetyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2,4-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrrole-3-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)butanamide
4-(2-chloropyridine-4-carbonyl)-6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
1-(4,4-difluoropiperidin-1-yl)-2-(2,3-dihydro-1H-inden-1-yl)ethan-1-one
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2-(1H-pyrazol-1-yl)benzamide
2-[2-amino-6-(dimethylamino)pyrimidin-4-yl]benzamide
1-{[2-(5-methylfuran-2-yl)phenyl]methyl}-4-(1H-pyrazol-3-yl)piperidine
2-(2-methyl-1,3-thiazol-4-yl)-5-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}pyrimidin-4-ol
2-(aminomethyl)-N-[2-(3-methylphenyl)-1,3-benzoxazol-6-yl]morpholine-4-carboxamide
1,3-dimethyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-cyclobutyl-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
{1-[(6-methoxy-2H-chromen-3-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
3-[4-(benzyloxy)piperidine-1-carbonyl]-1-methylpiperidine
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(3-phenylbutyl)-1,4-diazepan-5-one
4-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-ethylfuran-2-carboxamide
3-[({1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
2-benzyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,3-thiazole-4-carboxamide
N-methyl-6-(oxolan-3-ylmethyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-(2-chlorophenyl)-4-[(4-methoxy-3-{[1-(4-methylbenzoyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
2-(2-oxo-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-1,2-dihydroisoquinolin-1-one
1-methyl-4-{3-[1-(4,4,4-trifluorobutyl)-1H-pyrazol-3-yl]phenyl}-1H-pyrazole
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
1-cyclopropanecarbonyl-3-[2-(4-fluorophenyl)ethyl]piperidine
2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-3-(piperidine-1-carbonyl)pyrazine