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(2R,4R)-N-[2-(4-fluorophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide
1-[(3-methoxyphenyl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-N-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
8-chloro-2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
N-[3-(furan-2-yl)propyl]quinoxaline-6-carboxamide
benzyl({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-{1,4-diazabicyclo[3.2.2]nonan-4-yl}-N-(2-methoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-(propan-2-yl)-3-(pyridin-4-yl)propanamide
methyl 6-[2-(2,5-difluorophenyl)acetyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(2-chlorophenyl)-2-hydroxy-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
4-benzyl-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]acetamide
4-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-methylphenyl)acetamide
1-[(3-methylpyridin-2-yl)methyl]-4-[4-(piperidin-3-yl)benzoyl]piperazine
1-(cyclobutylmethyl)-3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}piperidin-2-one
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(3-methoxyphenyl)-1H-indazol-1-yl]acetamide
3-[1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-(carbamoylmethoxy)-N-[(2-methoxyphenyl)methyl]-N-propylbenzamide
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)amino]pyridine-3-carbonitrile
(3S,4R)-N,N-dimethyl-1-[(3-methylquinoxalin-2-yl)methyl]-4-propylpyrrolidin-3-amine
5-[(1E)-pent-1-en-1-yl]-1H-indazol-3-amine
1-{6-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]pyrimidin-4-yl}piperidin-4-ol
3,5-difluoro-N-(1-hydroxybutan-2-yl)-N-[(2-methylphenyl)methyl]pyridine-2-carboxamide
3-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}pyridin-2-amine
4-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-6-(methoxymethyl)pyrimidine
2-[4-(1-benzylpiperidin-4-yl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
2-ethyl-8-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
N-[4-(furan-2-yl)phenyl]-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine-3-carboxamide
N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-cyclopropyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,4-triazole
6-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
methyl 2-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetate
6-(3-chlorophenyl)-N-(cyclopropylmethyl)-N-propylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[3-(1H-imidazol-1-yl)propyl]-2-(3-methylthiophen-2-yl)-1H-imidazole
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-methylpyridine-3-carboxamide
3-[({1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
1-(oxane-4-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
3-ethyl-1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine
2-(oxolan-2-ylmethyl)-9-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)butanamide
8-[(2-carboxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)benzoic acid
1-benzyl-4-[3-(trifluoromethyl)pyridin-2-yl]-1,4-diazepan-6-ol
2-methyl-1-[2-(phenylsulfanyl)acetyl]-1,4-diazepan-5-one
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-6-ethoxyphenol
N-(cyclopropylmethyl)-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-N-propyl-1H-pyrazole-4-carboxamide