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5-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
(3R,4R)-1-(3-fluoropyridin-4-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-(2,6-dimethylphenyl)-2-[2-(1H-1,2,4-triazol-1-yl)propanamido]benzamide
4-(2-chlorophenoxy)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidine
2-(3-phenylpropyl)-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]morpholine
4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
4-benzyl-1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-N-methylpyridine-4-carboxamide
2-({4-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-1,3-benzothiazole
1-phenyl-4-(1-phenyl-1H-pyrazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2S,4R)-4-{[(5-chloro-2-hydroxyphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
N-methyl-2-(1-methyl-1H-imidazol-2-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-(4-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-3,5-dimethyl-1H-pyrrol-2-yl)ethan-1-one
4-(1H-pyrazol-1-yl)-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidine
N-methyl-2-(5-methyl-1H-pyrazol-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-(1-ethylpiperidin-4-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
3,5-dimethyl-4-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-1,2-oxazole
2-cyclobutaneamido-N-[2-(methylsulfanyl)ethyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-methyl-8-[1-(methylsulfanyl)propan-2-yl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-fluoro-2-methylphenyl)ethan-1-one
4-(azocan-1-yl)-N-(2-hydroxyethyl)-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
methyl(3-{2-[3-(1H-pyrazol-3-yl)phenyl]phenoxy}propyl)amine
4-[1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1H-imidazol-2-yl]pyridine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-(4-methoxyphenyl)furan-2-carboxamide
1-[(1-ethyl-1H-indol-6-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-methyl-2-(methylamino)-2-(thiophen-2-yl)-N-(thiophen-3-ylmethyl)acetamide
3-ethyl-3-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-(5-fluoropyridin-3-yl)urea
1-[2-(dimethylamino)ethyl]-N-[(5-fluoro-1H-indol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-ethyl-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
4-{2-[(6-ethylpyrimidin-4-yl)oxy]hex-5-en-1-yl}thiomorpholine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N,1-dimethyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
8-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)-2,8-diazaspiro[4.5]decan-3-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(piperidin-1-yl)acetamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{[(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-[(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)amino]propane-1,2-diol
3-(4-methoxy-2-methylbenzoyl)-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
8-(1-methyl-4-phenylpiperidine-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-fluoropyridine
2-(1-cyclopentyl-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-benzyl-7-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinoline-2-sulfonamide
2-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}quinolin-8-ol
2-(cyclopentylmethyl)-6-methyl-4-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3-carboxamide
N-methyl-5-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-[(1-cycloheptylpiperidin-4-yl)oxy]-N-cyclopropyl-4-methoxybenzamide
1-{[1-(6-{methyl[2-(methylamino)ethyl]amino}pyridine-3-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one