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N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3-chloro-N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzamide
4-[(3aS,6aS)-1-(1H-imidazol-4-ylmethyl)-octahydropyrrolo[2,3-c]pyrrol-5-yl]-5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidine
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
N-[3-(1H-indol-2-yl)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-3-carboxamide
2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1-(pyrrolidin-1-yl)ethan-1-one
2-[(4-ethoxypyrimidin-2-yl)amino]-1-(pyridin-3-yl)ethan-1-ol
3-hydroxy-3-{[(3-hydroxy-2,2-dimethylpropyl)amino]methyl}-1-[(3-methoxyphenyl)methyl]piperidin-2-one
4,6-dimethyl-2-oxo-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1,2-dihydropyridine-3-carboxamide
5-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N-methylpyrimidin-2-amine
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-6-methoxyphenol
(cyclohex-3-en-1-ylmethyl)({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(1H-imidazol-4-yl)ethyl]pyrimidine-5-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(1H-pyrazol-3-yl)piperidine
1-benzyl-N,N-dimethyl-5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
6-{[(2S,5R)-5-{[ethyl(methyl)amino]methyl}oxolan-2-yl]methyl}-3-methyl-1,2,3,4-tetrahydroquinazolin-2-one
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-5-methoxy-4H-pyran-4-one
3-fluoro-N-[1-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
1-[(4-chlorophenyl)methyl]-5-[4-(methoxymethyl)piperidine-1-carbonyl]piperidin-2-one
4-[(2S,4R)-1-(cyclohexylmethyl)-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
N-[4-(2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethoxy)phenyl]propanamide
2-methyl-6-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]pyrimidin-4-ol
2-(1-{[1-(9H-purin-6-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-[4-(benzyloxy)piperidin-1-yl]-2-(dimethyl-1H-1,2,4-triazol-1-yl)ethan-1-one
(3S,4S)-4-cyclopropyl-1-(oxan-4-ylmethyl)pyrrolidine-3-carboxylic acid
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-(1,4-dioxan-2-ylmethyl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
9-[(2E)-2-methylbut-2-en-1-yl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}-N-(pyridin-3-ylmethyl)benzamide
N-[(3S)-1-benzylpyrrolidin-3-yl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-[2-(azocane-1-carbonyl)morpholin-4-yl]-3-(pyridin-3-yl)propan-1-one
8-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3-fluorophenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-(thiophen-2-ylmethyl)piperidine
1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-(1-cyclohexyl-1H-pyrazol-5-yl)urea
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-butylacetamide
1-acetyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]piperidine-4-carboxamide
7-[3-(1H-pyrazol-1-yl)phenyl]-1,2,3,4-tetrahydroisoquinoline
3-fluoro-4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
5-(methoxymethyl)-N-(4-{5-methyl-4-[(3-phenylprop-2-ynamido)methyl]-1,3-oxazol-2-yl}phenyl)furan-2-carboxamide
1-{2-[(4aS,8aR)-2-oxo-1-propyl-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-{1-[2-(piperidin-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrazine
5-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-2-(pyridin-2-yl)pyrimidine