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3-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
N-[3-(4-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-(4-methylphenoxy)acetamide
(4aS,8aR)-6-(4-methoxypyrimidin-2-yl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-2-(methylsulfanyl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-(quinolin-5-ylmethyl)acetamide
8-[(2-aminopyridin-3-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-phenylacetamide
9-(5-methylpyrazine-2-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(azepane-1-carbonyl)piperidin-1-yl]-2-(3,4-dimethoxyphenyl)-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 2-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-2-yl]acetate
(3S,9aR)-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-(3-phenylpropyl)-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(furan-2-yl)ethyl]-1H-pyrazole-3-carboxamide
N-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
1-[3-(dimethylsulfamoyl)-5-[(naphthalen-1-ylmethyl)amino]benzoyl]piperidine-3-carboxamide
8-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(2S,4R)-1-[(3,4-difluorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
N-[(3S,4R)-1-(4-chloro-2-fluorobenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine
2-methoxy-N-[(3R,4S)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
6-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(4-methyl-1,4-diazepane-1-carbonyl)-6-azaspiro[2.5]octane
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
ethyl 6-[3-(4-fluorophenyl)pyrrolidin-1-yl]pyridine-3-carboxylate
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-7-methoxyquinolin-2-ol
4-(methoxymethyl)-1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine
(3S,4S)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(4-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
1-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)propan-1-one
2-amino-4-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-(dimethylamino)-2-(4-fluorophenyl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}acetamide
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(4-{[2-methoxy-2-(thiophen-2-yl)ethyl]amino}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
2-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl N-[(3S,5S)-5-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]carbamoyl}-1-methylpyrrolidin-3-yl]carbamate
(3aR,6aS)-5-{[2-(4-methoxyphenyl)ethyl]carbamoyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-(2-{[1-(4-methoxyphenyl)piperidin-4-yl]amino}ethyl)-N-methylmethanesulfonamide
N-[3-({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}sulfamoyl)phenyl]acetamide
1-(cyclobutylmethyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
N-{1-[4-(piperidin-3-ylmethyl)benzoyl]piperidin-4-yl}pyridin-2-amine
N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-4-(propan-2-yl)-1,2,3-thiadiazole-5-carboxamide
8-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
N-propyl-2-[3-(1H-pyrazol-3-yl)phenyl]benzamide
1-ethyl-4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
5-oxo-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide