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N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(pyrimidin-5-yl)pyridine-3-carboxamide
3-(1-ethyl-1H-pyrazol-3-yl)-4-[(2-fluorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(4aS,7aR)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-4-amine
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-yl]urea
1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(pyridin-3-yl)propan-1-one
(2S,4S,5R)-5-(2-chlorophenyl)-4-[(2-hydroxyethyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylic acid
(2R,6R)-4-(2-methoxy-6-methylbenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(1-methylpiperidin-2-yl)methyl]-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]ethan-1-one
2-(dimethyl-1,2-oxazol-4-yl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
7-(4-methoxypyrimidin-2-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
1-[1-(cyclopropylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
N'-[(2-ethoxyphenyl)methyl]-N,N-dimethyl-N'-(prop-2-en-1-yl)butanediamide
7-(2,3-dimethoxyphenyl)-9-methoxy-4-[(5-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2-(trifluoromethyl)benzamide
5-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyrimidin-2-amine
(4-{[1-(1-ethylpiperidin-4-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-{9-[(5-methylfuran-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyridin-4-yl)ethan-1-one
8-(cyclohex-3-en-1-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2E)-3-(3,5-difluorophenyl)prop-2-enoyl]-4-ethyl-1,4-diazepan-5-one
4-[4-(4-phenylpiperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-hydroxy-N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
4-methanesulfonyl-2-{[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}morpholine
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(oxolan-3-ylmethyl)amine
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-(2,3-difluorobenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N'1-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N'1-(oxolan-2-ylmethyl)cyclopropane-1,1-dicarboxamide
5-chloro-2-methoxy-N-methyl-N-(quinolin-5-ylmethyl)benzamide
4-({4-methyl-5-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
2-(5-methyl-1,2-oxazol-3-yl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)pyrrolidine-1-carboxamide
2-[(4aS,7aR)-6,6-dioxo-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
4-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-N-methyl-1,3-thiazol-2-amine
2-(4-fluorophenyl)-3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-6-methylquinoline
3-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]urea
5-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-cyclopropyl-8-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-ethyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)piperidin-4-amine
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]pyridin-2-amine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(2-oxopyrrolidin-1-yl)acetamide
{2-[3-(cyclopropylmethyl)-1-(4-methylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}dimethylamine
propan-2-yl 4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
N-(2-tert-butylphenyl)-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine-1-carboxamide
1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
1-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
(3aS,6aS)-2-(ethanesulfonyl)-5-(quinolin-6-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid