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methyl 2-(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
6-methyl-5-[5-(1-methyl-4-phenylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-[2-(dimethylamino)ethyl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-ethyl-5-[3-(2-ethylphenoxy)azetidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-(2-methylphenyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-ol
2-cyclobutaneamido-N-(3-ethoxypropyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
[4-(oxan-2-ylmethyl)-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl]methanol
4-(1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-imidazol-2-yl)-2,1,3-benzoxadiazole
2-{4-[6-methyl-2-(methylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}-N-[1-(2-methylpropyl)-1H-pyrazol-5-yl]acetamide
3-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]propanoic acid
(1-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-oxooxolan-3-yl)acetamide
N-[(1-{[4-(pyridin-2-yl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
1-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-3-phenyl-1H-pyrazole-5-carboxamide
8-(dimethyl-1,3-oxazole-5-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-chloro-2-[2-(3-methoxypropyl)piperidine-1-carbonyl]-1H-indole
[4-benzyl-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]methanol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]butan-1-one
N-[(2-methoxyphenyl)methyl]-4-methyl-N-(prop-2-en-1-yl)piperidine-4-carboxamide
2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(oxan-2-ylmethyl)acetamide
1-{4-[2-(quinolin-2-yloxy)hex-5-en-1-yl]piperazin-1-yl}ethan-1-one
(3S,4S)-1-(3-chloro-4-methoxybenzoyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
(3R,4R)-3-cyclobutyl-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-4-methylpyrrolidin-3-ol
2-(5-acetylthiophen-3-yl)-N-[1-(1H-indol-5-yl)ethyl]acetamide
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-3-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
2-methyl-5-(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1,3,4-oxadiazole
3-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}pyridin-1-ium-1-olate
2-[4-methyl-6-(4-{[(5-methyl-1H-imidazol-4-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-yl]phenol
4-(1H-1,3-benzodiazol-2-ylmethyl)-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-[2-(dimethylamino)-1-phenylethyl]-2-(hydroxymethyl)-N-methyl-1H-1,3-benzodiazole-5-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-ol
N-(2-fluoroethyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-cyclooctyl-2-({[(2S)-5-oxopyrrolidin-2-yl]methyl}(pyridin-4-ylmethyl)amino)acetamide
2-[4-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethan-1-ol
(2S,4S)-4-[4-(4-fluoro-2-methylbenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-methyl-4-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}pyrimidine
5-ethyl-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-(1-methylpyrrolidin-3-yl)-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
N-(3-methylphenyl)-3-[(1,2-oxazol-3-ylmethyl)sulfamoyl]benzamide
3-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)-5-methoxy-1H-indazole
N-[3-(4-methoxyphenyl)propyl]-6-{pyrazolo[1,5-a]pyridin-7-yl}pyridine-3-carboxamide
1-[2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]imidazolidin-2-one
4-methyl-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperidine
(4aS,8aS)-2-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-decahydro-2,7-naphthyridin-4a-ol
1-(4-benzylpiperidin-1-yl)-3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]propan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
5-[({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-(4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole