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3-[1-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-8-fluoro-3,4-dihydroquinazolin-4-one
[2-(4-methoxy-3,5-dimethylphenyl)phenyl]methanamine
N-ethyl-6-[(1E)-pent-1-en-1-yl]pyridine-3-carboxamide
2-methyl-5-(3-phenylpiperazine-1-carbonyl)pyrimidine
2-{1-[(4-ethoxyphenyl)methyl]-4-(1H-indol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N1,N1-dimethyl-N4-{2-[(3-methylpyridin-2-yl)amino]ethyl}piperidine-1,4-dicarboxamide
2-methoxy-N-(1-{4-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
3-[({1-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperidin-3-yl}oxy)methyl]pyridine
benzyl 4-(2-ethylpyrimidine-5-carbonyl)-1,4-diazepane-1-carboxylate
N-(2,3-dihydro-1H-inden-2-yl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(2-methoxyethyl)-3-{[2-(2-methylphenyl)-1H-imidazol-1-yl]methyl}-4H-1,2,4-triazole
3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
4-methyl-6-[4-(oxolane-2-carbonyl)piperazin-1-yl]-2-propylpyrimidine
N-{[1-(1H-indol-2-ylmethyl)pyrrolidin-3-yl]methyl}-4-methylpyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-(2-{3-[1-(dimethylamino)ethyl]phenyl}-4-fluorophenyl)ethan-1-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]azepan-4-amine
2-(2-methoxyethyl)-N-(2-phenoxyphenyl)morpholine-4-carboxamide
1-[(8-methoxy-2H-chromen-3-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
N-[(5-methylthiophen-2-yl)methyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-[2-(2-oxo-5,5-diphenylpiperidin-1-yl)ethyl]-1,3-oxazinan-2-one
3-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-[(1S,5R)-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-(5-methylthiophen-2-yl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
2-[(dimethylamino)methyl]-N-[5-methoxy-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,3-thiazole-4-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-7-methyl-2,7-diazaspiro[4.4]nonane
6-methoxy-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]hexan-1-one
1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-3-(1H-pyrazol-3-yl)piperidine
N-[2-({[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]carbamoyl}amino)ethyl]pyridine-3-carboxamide
4-(2-fluoroethyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N3-methyl-1-(3-methylbutyl)-4-oxo-N5-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N,N-dimethyl-2-[(1S,5R)-3-[2-(methylsulfanyl)benzoyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
5-cyclopropyl-N-ethyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
1-[(6-ethylpyrimidin-4-yl)amino]-3-(pyrrolidin-1-yl)propan-2-ol
3-(3-hydroxy-3-methylbutyl)-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)benzamide
3-cyclopropyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
2-ethyl-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-methyl-4-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}benzene-1-sulfonamide
4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-8-thia-4,6-diazatricyclo[7.6.0.02,7]pentadeca-1(9),2(7),5-trien-3-one
3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
7-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-4-methyl-2H-chromen-2-one
(3aS,6aR)-5-(3-methylfuran-2-carbonyl)-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
[(4aS,8aR)-6-{[3-(pyridin-2-yl)phenyl]methyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
2-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-4-amine
5-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-4,6-dimethyl-2H-pyran-2-one
1-{1-[(3-fluorophenyl)methyl]piperidin-3-yl}-4-phenylpiperazine