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2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-phenylacetamide
1-(pyridin-3-ylmethyl)-4-[4-(2,2,2-trifluoroethyl)piperazine-1-carbonyl]pyrrolidin-2-one
7-methoxy-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 4-{[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}-1H-pyrazole-3-carboxylate
4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
2-ethyl-8-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-2,3-dihydro-1H-isoindole
4-[(2,5-dimethylthiophen-3-yl)sulfonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
8-(3-hydroxy-2-methylbenzoyl)-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1,3-dimethyl-4-({2-[(4-methylphenyl)methoxy]phenyl}methyl)piperazin-2-one
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-(butan-2-yl)-5-(2-methoxypyridin-3-yl)furan-2-carboxamide
3-[benzyl({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})amino]-1λ6-thiolane-1,1-dione
2-(dimethylamino)-7-(2-propyl-1,3-thiazole-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-[3-(1H-indol-3-yl)propanoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyrazine
(2R,3R,6R)-3-(2-methoxyphenyl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 3-[2-(morpholin-4-yl)-6-oxo-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-8-yl]benzoate
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
(1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-3-yl)methanol
9-(3-ethyl-1H-pyrazole-5-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-2-(pyridin-3-yl)pyrimidin-4-amine
1-cyclohexyl-1-methyl-3-[3-(1,3-oxazol-5-yl)phenyl]urea
4-{5-[(dimethyl-1,3-thiazol-5-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridine
3,5-dimethyl-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-1,2-oxazole-4-sulfonamide
1-(furan-3-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-1-(4-fluorophenyl)butan-1-one
3-[5-(3-chloro-4-methylbenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-{2-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}phenol
2-{[1-(4-methyl-1,4-diazepane-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]methyl}-1,3-benzothiazole
N,2-dimethyl-3-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)propanamide
(4S)-3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
2-(2,3-dihydro-1-benzofuran-7-yl)-2-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}acetic acid
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[methyl(propan-2-yl)amino]methyl}phenoxy)propan-2-ol
(1R,5S,8S)-3-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
4-(6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-yl)morpholine
2-methyl-5-{2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
3-(1-{[2,5-dimethyl-1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}piperidin-4-yl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[1-benzyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-methyl-1-(1,4-oxazepan-6-ylmethyl)-3-phenylurea
methyl (1R,5S,6R)-6-{[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
1-(2-methoxyethyl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine-3-carboxamide
1-(3,5,7-trimethyl-1H-indole-2-carbonyl)azetidine-2-carboxylic acid
ethyl 1-[1-(propan-2-yl)piperidin-4-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3-{1-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-pyrazol-4-yl}benzoic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-cyclohexylpiperidin-3-ol