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N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(2-methylpyridin-3-yl)oxy]-N-(propan-2-yl)piperidine-4-carboxamide
(1R,3S)-3-amino-N-[(4-fluorophenyl)methyl]-N-(pyridin-4-ylmethyl)cyclohexane-1-carboxamide
N-[1-(methoxymethyl)cyclopentyl]-5,6-dimethylpyridine-3-carboxamide
5-(3-methylbut-2-en-1-yl)-1'-(oxolan-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
({3-[(dimethylamino)methyl]phenyl}methyl)[1-(2,6-dimethylphenoxy)propan-2-yl]amine
2-ethoxy-6-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}phenol
methyl 4-(4-{[(1,3-benzothiazol-2-ylmethyl)(methyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
1-methyl-8-[2-(2-methyl-1H-indol-3-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(propan-2-yl)-1-[1-(quinoline-6-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
N-[4-(4-{[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}piperidin-1-yl)phenyl]-3-phenylpropanamide
2-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]-2-azabicyclo[2.2.1]heptane
N-[1-(1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-2-phenylethyl]-N-methylpyridine-2-carboxamide
1-(4-cyclopentylpiperazin-1-yl)-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-methyl-N-(pyridin-3-ylmethyl)pyridin-2-amine
N-ethyl-6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxamide
8-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{2-oxo-2-[2-(pyridin-3-yl)piperidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
2-(dimethylamino)-N-(3-methyl-1-{7-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
2-[3-({[2-(azepan-1-yl)ethyl](ethyl)amino}methyl)phenoxy]acetamide
{imidazo[1,2-a]pyridin-3-ylmethyl}({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
2-amino-4-(5-ethylfuran-2-yl)-6-(2-methylpropanoyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2,2-dimethyl-N-(1-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-4-(thian-4-yl)piperazine
N-(3-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
2-methyl-5-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}phenol
3-[5-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
(1S,5R)-3-methyl-6-(6-methylpyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-fluorophenyl)-3-[1-(thiophene-3-carbonyl)piperidin-3-yl]propanamide
6-fluoro-3-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]quinolin-4-ol
3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
7-[(2,5-dimethylthiophen-3-yl)sulfonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-3,4,7-trimethyl-1H-indole
7-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(2S)-1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-oxopropan-2-yl]acetamide
3-(1H-imidazol-2-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}benzamide
(1R,6S)-9-methyl-3-[2-(morpholine-4-carbonyl)pyridin-4-yl]-3,9-diazabicyclo[4.2.1]nonane
8-fluoro-3-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}phenol
5-[(4-methoxyphenyl)methyl]-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methoxy-5-{[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenol
(3S,4R)-1-(2-amino-2-methylpropanoyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-(2,6-difluorophenoxymethyl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
6,7-dimethoxy-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2,3,4-tetrahydroisoquinoline
6-fluoro-3-[2-(2-hydroxyethoxy)ethyl]-3,4-dihydroquinazolin-4-one