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4-{1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]azetidin-3-yl}pyridine
N-[4-(4-butyl-3-oxopiperazine-1-carbonyl)phenyl]cyclobutanecarboxamide
[(3R,4R)-1-(benzenesulfonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-4-propylpyrimidine-5-carboxamide
1-{2-[4-(2-phenylethyl)piperazin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
4-{5-[1-(1H-imidazol-1-yl)ethyl]-3-methyl-1H-1,2,4-triazol-1-yl}-2-methylpyridine
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}quinoline-8-sulfonamide
4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
1-(cyclohexylmethyl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-6-oxopiperidine-3-carboxamide
3-(5-methylfuran-2-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrazole-5-carboxamide
5-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
N-(2-methylpropyl)-1-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-(2-methoxyethyl)-8-(5-methoxypyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
6-fluoro-2-oxo-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
7-cyclopentyl-2-[6-(methoxymethyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-6-(2-methoxyethyl)-3-{[2-(propylamino)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-4-(2-cyanobenzamido)-N-ethyl-1-[2-(methylsulfanyl)acetyl]pyrrolidine-2-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]propanamide
2-(2-methoxyethyl)-9-(2,4,5-trimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-hydroxycyclohexyl)methyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(2R,3R)-3-{[2-(1H-indol-3-yl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(1H-indol-5-ylmethyl)-1-[4-(oxan-2-ylmethoxy)phenyl]urea
6-methoxy-N-[2-(4-methylbenzenesulfonyl)ethyl]pyrimidin-4-amine
1-(1-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}azetidin-3-yl)-2-methylpiperidine
{1-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
3-[3-cyclopropyl-1-(4-methanesulfonylphenyl)-1H-1,2,4-triazol-5-yl]-1H-indazole
[(2S,6S)-4-(cyclopropylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(2S)-1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-hydroxy-3-phenylpropan-1-one
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
1-[(3,4-difluorophenyl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
5-[(1-benzylpiperidin-4-yl)amino]-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}acetamide
1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-methyl-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-1,3-thiazole-4-carboxamide
2-[N-(3-methylphenyl)methanesulfonamido]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-(2-methoxyethyl)-1-[3-(piperidine-1-carbonyl)pyridin-2-yl]piperidine-3-carboxylic acid
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(2-phenoxyethyl)piperazine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidine
2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-4-(oxolan-3-yl)-1H-1,2,3-triazole
6-fluoro-N-methyl-2-oxo-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-cyclobutyl-2-[3-(furan-2-yl)-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
2-(dimethylamino)-N-{[4-(dimethylamino)-1-ethylpiperidin-4-yl]methyl}-2-(2-fluorophenyl)acetamide
3-{2-oxo-2-[1-(pyridin-3-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl]ethyl}imidazolidine-2,4-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
5-({[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
1-[(3S,4R)-1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea