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1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-4-(piperidin-1-yl)butan-1-one
1-(1,2-oxazol-3-ylmethyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
3-[3-(1H-1,3-benzodiazol-2-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(butan-2-yl)-N-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]cyclopentanamine
2-{1-[2-(methylamino)pyrimidine-5-carbonyl]pyrrolidin-3-yl}benzoic acid
3-(3-methyl-1H-pyrazol-1-yl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]propan-1-one
methyl 3-{[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}propanoate
1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-(1H-pyrazol-5-ylmethyl)benzamide
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-4-(quinoxaline-5-carbonyl)-1,4-diazepan-2-one
3-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
6-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-{2-[(3-phenyl-1H-pyrazol-4-yl)formamido]ethyl}piperidine-3-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-6-ethylpyrimidin-4-amine
N-(2-methoxyethyl)-4-[(2-methylpyridin-3-yl)oxy]-N-propylpiperidine-4-carboxamide
1-[cyclohexyl(methyl)amino]-3-{3-[(4-ethyl-1,4-diazepan-1-yl)methyl]phenoxy}propan-2-ol
1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-4-[3-(propoxymethyl)pyrrolidin-1-yl]piperidine
2-(azepan-1-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
(1R,5R)-6-benzyl-3-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-methyl-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)piperidine-4-carboxamide
1-(6-chloroquinolin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(4-methoxybenzoyl)-4-(1H-pyrrole-3-carbonyl)piperazine
1-(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-3-methylbutan-1-ol
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]acetamide
4-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-6-methyl-2-propylpyrimidine
N-methyl-2-{5-[(2E)-pent-2-en-2-yl]-4-phenyl-1H-imidazol-1-yl}butanamide
2-{3-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
2-[3-(4-fluorophenyl)-4-methyl-1H-pyrazol-1-yl]-N-(2-propyl-2H-1,2,3-triazol-4-yl)acetamide
5-{3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl}-4-methylpyrimidin-2-amine
N,N-diethyl-5-[(E)-2-phenylethenyl]furan-2-carboxamide
2-methyl-9-[2-(pyrrolidin-3-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
4-(1-methyl-1H-indole-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-(1-benzyl-1H-pyrazol-3-yl)-2-(3,5-dimethyl-4-phenyl-1H-pyrazol-1-yl)acetamide
1-{5-[3-(5-methylfuran-2-yl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidine
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N4-{[2-(diethylamino)pyridin-3-yl]methyl}-N1,N1-dimethylpiperidine-1,4-dicarboxamide
N-(2-methoxyethyl)-2-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-benzofuran-5-carboxamide
3-(4-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-2-oxopiperazin-1-yl)benzonitrile
1-(2-{[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)amino}ethyl)piperidin-2-one
1-[4-(4-{6-[(thiophen-2-ylmethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperazin-1-yl)phenyl]ethan-1-one
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[4-(methylsulfanyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl 1-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]cyclopropane-1-carboxylate
5-methyl-N-[1-(thiophen-2-yl)propan-2-yl]-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-[2,2-bis(prop-2-en-1-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
4-{[1-(2-ethyl-1H-imidazol-1-yl)propan-2-yl]amino}-N-phenylpiperidine-1-carboxamide
2-(2,4-dimethoxyphenyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide