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1-(4-benzylpiperazin-1-yl)-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}propan-1-one
[(1-cyclohexylpiperidin-3-yl)methyl][(5-methylthiophen-2-yl)methyl](pyridin-3-ylmethyl)amine
4-[5-(1,2,3-thiadiazol-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
1-methyl-5-{[1-(3-phenylphenyl)piperidin-4-yl]amino}piperidin-2-one
2-(4-fluorophenyl)-2-hydroxy-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}acetamide
2-chloro-N-[2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylformamido)ethyl]benzamide
N-[1-(5-acetylpyridin-2-yl)piperidin-4-yl]methanesulfonamide
N-cyclopropyl-2-(2-methyl-1,3-thiazol-4-yl)-N-(1,3-thiazol-5-ylmethyl)acetamide
ethyl 4-(6-{[2-(furan-2-yl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carbonyl)piperazine-1-carboxylate
5-acetyl-6-methyl-3-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-(cyclopropylmethyl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
4-[1-(benzenesulfonyl)cyclopropanecarbonyl]piperazine-2-carboxylic acid
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-8-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(pyridine-2-carbonyl)piperidin-4-amine
N-(butan-2-yl)-3-(carbamoylmethoxy)-N-(pyridin-4-ylmethyl)benzamide
3-methanesulfonamido-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
(2S)-2-amino-N-ethyl-3-(4-hydroxyphenyl)-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
N-[3-chloro-4-(propylcarbamoyl)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
4-[1-benzyl-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
1-[(2-fluorophenyl)methyl]-N-[1-(pyridin-4-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
4-(quinolin-3-yl)-1H-pyrazole-3-carbonitrile
2-[5-(6,6-dimethyl-5-oxothiomorpholin-3-yl)-1-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl]acetamide
8-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl[(1-{[1-(9H-purin-6-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
2-(azocane-1-carbonyl)-4-chloro-1-methyl-1H-indole
N-cyclopropyl-4-hydroxy-N-[(3-methylthiophen-2-yl)methyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1-[(2-fluorophenyl)methyl]piperidin-3-amine
3-[(dimethylamino)methyl]-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
2-(2,3-difluorophenoxymethyl)-N-methyl-N-(oxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,3-dimethyl-5,6-dihydro-1,4-dioxine-2-carboxamide
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]propanamide
(1S,6R)-9-{3-azaspiro[5.5]undecan-9-yl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
5-(4-acetylphenoxymethyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[3-(morpholin-4-yl)propyl]propanamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-methyl-2-(methylamino)-1,3-thiazole-5-carboxamide
2-{2-[4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-1,2,3-triazol-1-yl]propyl}-3-methylpyridine
methyl 2-({2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}amino)acetate
1-(3-cyanobenzoyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-(butan-2-yl)-3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
5-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
2-[1-(1,1-dioxo-1λ6-thiolan-3-yl)-4-phenyl-1H-imidazol-5-yl]benzoic acid
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)amine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyrrolidin-1-yl)propan-1-one
8-fluoro-2-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)quinolin-4-ol
3-ethyl-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1H-indole
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
3-{[(3S,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}-7-methyl-1,2-dihydroquinolin-2-one