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3-cyclopentyl-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
(2E)-3-(2,3-difluorophenyl)-1-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)prop-2-en-1-one
N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2R)-2-{[3-ethoxy-4-(prop-2-en-1-yloxy)phenyl]formamido}propanamide
1-[4-(2-amino-4-phenylpyrimidine-5-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
(dicyclopropylmethyl)({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-(pyridin-2-yl)propan-1-one
(2R,6R)-4-(1-ethyl-1H-pyrazole-5-carbonyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-benzyl-3-ethyl-1-(1-methyl-1H-indazole-3-carbonyl)-1,4-diazepan-5-one
5-[4-(2-ethoxyphenyl)piperazin-1-yl]-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-cyclohexanecarbonyl-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[3-(hydroxymethyl)benzoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
5,6-dimethoxy-2-(1,3-thiazol-4-ylmethyl)-1,2-dihydroisoquinolin-1-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine-2-carboxamide
1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
4-[(4-methyl-5-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
5-{[2-(8-chloroquinolin-2-yl)-1H-imidazol-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
6-ethyl-N4-(1-ethylpiperidin-3-yl)-N2,N2-dimethylpyrimidine-2,4-diamine
2-(6-methoxynaphthalen-2-yl)-4-(1H-pyrrole-3-carbonyl)morpholine
5-{[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)propanamide
1-[1-(methoxymethyl)cyclopropanecarbonyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
(2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)urea
4-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1λ6-thiomorpholine-1,1-dione
2-({3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}methyl)phenol
5-methoxy-2-({4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
2-(2,2-dimethylpropanamido)-N-[2-(1H-imidazol-4-yl)ethyl]-5-methylthiophene-3-carboxamide
1-[(4-fluorophenyl)methyl]-3-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]benzene-1-sulfonamide
6-(cyclopropylamino)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-(4-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}piperazin-1-yl)ethan-1-one
2-methyl-6-[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-3-yl]pyrimidin-4-ol
ethyl 3,5-dimethyl-4-{methyl[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]carbamoyl}-1H-pyrrole-2-carboxylate
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidine
N-{[7-(methylsulfanyl)-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
3-[5-(2,3-dihydro-1H-inden-1-ylmethyl)-1,2,4-oxadiazol-3-yl]pyridazine
5-{3-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
1-butyl-4-(2,5-dimethylphenyl)-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
2-[(2-chlorophenyl)methyl]-4-{4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]acetamide
4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}morpholine-2-carboxamide
2-{2-[5-(1-ethyl-1H-indol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethoxy}ethan-1-ol
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-3-[2-(morpholin-4-yl)pyridin-3-yl]-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
4-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}benzamide