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methyl 1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
2-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
ethyl 4-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-amido}piperidine-1-carboxylate
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-2-(1H-pyrazol-1-yl)acetamide
5-[({[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-(3-hydroxypropyl)-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
9-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,9aR)-1-(2-methylphenoxymethyl)-octahydro-1H-quinolizine
[(3S,5S)-1-(2H-1,3-benzodioxol-5-ylmethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
methyl({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl})(oxan-2-ylmethyl)amine
N3-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-1,3-dicarboxamide
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-4-(methoxymethyl)-5-methyl-1,2-oxazole
4-(4H-1,2,4-triazol-4-yl)-N-(2,2,2-trifluoroethyl)benzamide
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-6-yl]oxy}acetamide
8-(2-fluorobenzoyl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[2-amino-6-(methylamino)pyrimidin-4-yl]-N,N-bis(propan-2-yl)benzamide
5-{imidazo[1,2-a]pyridine-2-carbonyl}-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[4-(4-benzylpiperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-methyl-4-phenyl-5-(2,4,5-trimethoxyphenyl)-1H-imidazole
N-(3-hydroxy-1-oxo-1-{4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}propan-2-yl)acetamide
1-(2-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
5-(cyclobutylmethyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-{[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]amino}-N-(pyrazin-2-yl)acetamide
[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl][1-(morpholin-4-yl)propan-2-yl]amine
methyl (2S,3R)-2-[(3,5-dimethyladamantan-1-yl)formamido]-3-hydroxybutanoate
N-[(8-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}quinolin-3-yl)methyl]cyclopentanamine
(3R,4R)-1-{[5-(2,3-dichlorophenyl)furan-2-yl]methyl}-4-(hydroxymethyl)piperidin-3-ol
3-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-4-(3-methylbutyl)piperazin-2-one
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
1-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-{5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}pyrimidin-2-amine
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(pyrrolidin-3-yl)benzamide
2-(5-methyl-1-phenyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(3,4-dimethoxyphenyl)methyl]-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl][(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
N,2,6-trimethyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrimidine-4-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
N-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
1-{4-[(propan-2-yl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(3S,7S)-5-[3-(piperidin-1-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-[(4-cyanophenyl)methyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{4-[(2-chlorophenyl)methyl]-5-oxo-1,4-diazepan-1-yl}-2-phenylethane-1,2-dione
N-(2,3-dihydro-1H-inden-2-yl)-5-acetamido-2-hydroxy-N-methylbenzamide
4-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-4-oxo-N-phenylbutanamide