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1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aS,7aR)-1-(dimethyl-1,3-oxazole-4-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(5-phenoxyfuran-2-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
2-methyl-5-(4-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
N-[(2-fluorophenyl)methyl]-4-{4-[(thiophen-2-ylmethyl)amino]piperidin-1-yl}benzamide
propyl 8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
ethyl 4-{4-[1-(N-methyl-1-thiophen-2-ylformamido)-2-phenylethyl]piperidin-1-yl}piperidine-1-carboxylate
1-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxylic acid
(4aR,7aS)-1-(2-methoxyacetyl)-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-methylphenyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}piperidin-4-ol
1-(carbamoylmethyl)-N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}piperidine-4-carboxamide
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
1-ethyl-3-methyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
2-(3,4-dimethylphenoxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
2-[5-(thiomorpholine-4-carbonyl)-1H-pyrazol-3-yl]phenol
2-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]benzoic acid
2-{[(2S,4S)-4-[(4-fluorophenyl)sulfanyl]-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}phenol
3-{5-[3-(1-methyl-1H-pyrrol-2-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
6-methoxy-1-methyl-2-{3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}-1H-indole
(2S)-2-amino-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-amine
methyl 3-(cyclohex-3-en-1-ylmethyl)-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(3R,4S)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(piperidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
3-{2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-2-yl]ethyl}phenol
(3S,4R)-4-(2-methoxyphenyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidine-3-carboxylic acid
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2-fluorophenyl)methyl]piperidine
N-[1-(1H-indol-5-yl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyridine
2-amino-4-{2-[2-(dimethylamino)ethoxy]phenyl}-6-(furan-2-yl)pyridine-3-carbonitrile
methyl 3-{methyl[(1-phenylpyrrolidin-3-yl)methyl]carbamoyl}benzoate
5-{2-[(2-methoxyethyl)amino]ethyl}-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-one
6-[(diethylamino)methyl]-N-[2-(1,3-thiazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3H,4H-pyrido[4,3-d]pyrimidin-4-one
3-(1-benzothiophen-3-yl)-1-methyl-6-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(2,6-dimethylpyridin-3-yl)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carboxamide
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-4-fluoro-2-hydroxybenzamide
1-[3-(1H-imidazol-2-yl)benzoyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
1-cyclopentyl-4-[4-(difluoromethoxy)benzoyl]-1,4-diazepane
2-(dimethylamino)-N-[2-methyl-5-({[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)phenyl]acetamide
3-({[1-(5-ethyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]oxy}methyl)pyridine
4-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)-6-ethylpyrimidine
2-{2-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione
3-fluoro-5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
6-fluoro-2-oxo-N-[2-(pyridin-4-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(2-hydroxyphenyl)acetamide