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1-benzyl-3-(2-methoxyphenyl)-6-[3-(pyridin-2-yl)propanoyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(3S,4R)-1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-[3-(1H-pyrazol-1-yl)propyl]-1,3-oxazole-4-carboxamide
3-[4-(7-fluoro-4-methylquinolin-2-yl)piperazin-1-yl]propanamide
1-(2-chlorobenzenesulfonyl)-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
methyl 3-[(2,3-dimethoxyphenyl)methyl]-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-amino-6-methyl-N-(2-methylcyclohexyl)pyrimidine-4-carboxamide
(2S,4R)-4-(dimethylamino)-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidine-2-carboxylic acid
[(dimethyl-1,2-oxazol-4-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
3-{[3-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)piperidin-1-yl]methyl}phenol
4-[2-(3-methoxyphenoxy)ethyl]-3-methylpyridine
6-methyl-N4-[2-(2-methylpropanesulfonyl)ethyl]pyrimidine-2,4-diamine
8-(2-methyl-1,3-thiazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-(morpholin-4-ylmethyl)cyclopentan-1-amine
N-(4-methoxy-2-methylphenyl)-2-(morpholin-3-yl)acetamide
3-benzyl-7-[1-(4-chlorophenyl)cyclobutanecarbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-(6-methyl-2-phenyl-1,2-diazinane-1-carbonyl)-1,2-dihydroquinoxalin-2-one
N-{1-[3-cyclopentyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
1-cyclohexanecarbonyl-N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]pyrrolidine-2-carboxamide
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-6-methylpyridine-3-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl})amine
1-({5-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
methyl 6-[(oxolan-3-yl)amino]pyridine-3-carboxylate
2-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-1,2,3-triazol-4-yl)quinolin-4-ol
1-(2-methoxyphenyl)-N-(4H-1,2,4-triazol-4-yl)-1H-pyrazole-4-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
3-{2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
5-[1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-2-yl]-N-(4-hydroxybutyl)thiophene-2-carboxamide
N-cyclopropyl-3-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}propanamide
2-(4-{[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]methyl}phenyl)acetic acid
4-amino-3-hydroxy-1-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}butan-1-one
9-(1-aminocyclopropanecarbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzoic acid
N-[2-(dimethylamino)ethyl]-1-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydroisoquinoline-4-carboxamide
2-[N-(3-methylphenyl)methanesulfonamido]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]benzamide
5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amine
(4aS,8aR)-6-[(2-ethylpyrimidin-4-yl)methyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
N-cyclobutyl-3-[(3-ethoxy-2-hydroxypropyl)sulfamoyl]benzamide
2-(furan-3-yl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
2-[(4-chlorophenyl)methyl]-8-[(1-methylpiperidin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(2,3-dihydroxypropyl)-1-[4-(4-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-3-methylurea
1-[2-(4-chlorophenyl)ethyl]-5-[4-(propan-2-yl)piperidine-1-carbonyl]piperidin-2-one
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
6-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridine-3-carboxylic acid
methyl 6-(2-cyclopentylacetyl)-2-[(3,5-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate