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5-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)-1,3-benzoxazole
(3aS,6aS)-2-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}acetamide
2-(4-methoxyphenyl)-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}morpholine
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-propyl-1,2-oxazole-4-carboxamide
4-{1-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1H-imidazol-2-yl}-3-methoxyphenol
3-[(2-aminopyrimidin-5-yl)methyl]-1-(3-chloro-2-propoxyphenyl)-3-methylurea
2-(3-methoxypropyl)-9-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
4-[2-methyl-2-(piperidin-1-yl)propyl]-2-(pyridin-3-yl)morpholine
4-fluoro-3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]benzene-1-sulfonamide
3-(cyclopentylsulfamoyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
5-methyl-3-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-2-yl)-1,2-oxazole
(1R,5R)-6-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)[(3-methylpyridin-4-yl)methyl]amine
4-(2-fluorophenyl)-2-{5-methyl-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}pyrimidine
N-cyclopropyl-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carboxamide
6-[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2,3-dihydropyridazin-3-one
5-methyl-1'-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(3-fluorophenyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]acetamide
(furan-2-ylmethyl)(methyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
N-cyclopropyl-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
2-(3-methoxyphenyl)-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
1-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propan-1-one
4-methyl-6-(4-{[2-(pyridin-2-ylsulfanyl)ethyl]amino}piperidin-1-yl)pyrimidin-2-amine
propan-2-yl (1R,5S,6R)-6-{[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
(3aR,6aR)-2-(2-methoxyacetyl)-N-(1-phenylcyclopropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(3-methoxyphenoxymethyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
2-methyl-1-{1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}piperidine
methyl 4-(5-methyl-4-{[4-(morpholine-4-carbonyl)piperidin-1-yl]methyl}-1,3-oxazol-2-yl)benzoate
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(oxane-4-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
2-methyl-1-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}azetidin-3-yl)piperidine
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-chlorobenzamide
1-(1-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidin-3-yl)-1H-imidazole
N-(2-methoxyethyl)-1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-hydroxy-2-(pyridin-2-yl)ethyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
(3S)-1-{5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-methyl-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]quinolin-2-amine
2-{5-[(2-chlorophenyl)(hydroxy)methyl]-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
(1S,5R)-3-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}-2-(thiophen-3-yl)acetic acid
1-[(5-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
3-(2-ethylbutyl)-8-(1-methylpiperidine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}phenol
3-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-1-[(5-methylpyrazin-2-yl)methyl]urea
1-methyl-4-[3-(methylsulfanyl)propanoyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3-fluorophenyl)methyl]-3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
(3R,5S)-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
dimethyl(2-{4-[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperazin-1-yl}ethyl)amine