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5-{[(4aS,7aR)-4-(dimethylcarbamoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
[1-(ethylsulfanyl)propan-2-yl]({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
1-(4,6-dimethylpyrimidin-2-yl)-4-(piperidin-1-yl)piperidine-4-carboxamide
3-cyano-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]benzamide
(4aR,7aS)-4-(1-ethyl-1H-pyrazole-3-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(1-ethyl-1H-1,2,4-triazol-3-yl)-3-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]urea
1-(1,4-dioxane-2-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
methyl 5-[(4-methoxy-4-methylpentan-2-yl)amino]-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(adamantan-1-yl)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]acetamide
N-(furan-2-ylmethyl)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[2-(azepan-1-yl)-2-phenylethyl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
N-ethyl-2-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]benzamide
(4R)-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,3-dimethyl-1,3-thiazolidine-4-carboxamide
(3R,4S)-4-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
1-(5-chloro-2-methoxyphenyl)-5-(2-ethoxyethyl)-3-methyl-1H-1,2,4-triazole
2-({5-[2-(2-hydroxyphenyl)ethyl]-4-phenyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-benzyl-4-(3-methoxybenzoyl)piperazine-1-sulfonamide
5-phenyl-N-[2-(1,3-thiazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
5-fluoro-4-(morpholin-4-yl)-N-[1-(oxan-4-yl)piperidin-4-yl]pyrimidin-2-amine
6-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
4-phenyl-N-({1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-3-yl}methyl)benzamide
8-[(2-methoxypyridin-3-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
6-[4-(1-methoxyethyl)phenyl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-methyl-2-oxo-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-dihydropyridine-3-carboxamide
5-(3-fluorophenoxymethyl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-1H-pyrazole-3-carboxamide
1-[4-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
4-(1-hydroxy-2-{[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)phenol
1-{4-[1-cyclohexyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}-1H-1,2,3,4-tetrazole
4-(4-methoxyphenyl)-6-(6-methylpyridine-3-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
2-(dimethylamino)-N-{2-[(4-fluorophenyl)formamido]ethyl}-2-(2-methylphenyl)acetamide
(5S,9aS,9bS)-5-(4-hydroxy-3,5-dimethylphenyl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N,N-dimethyl-3-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]sulfamoyl}benzamide
1-(2-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}ethyl)pyrrolidin-2-one
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-propoxypiperidine
2-methoxy-4-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
N-[(4-methoxy-3-methylphenyl)methyl]-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
3-(azocan-1-yl)-N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]propanamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-benzyl-N-methyl-1,3-oxazole-4-carboxamide
N5-methyl-N5-[(1-methyl-1H-imidazol-2-yl)methyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-methyl-2-oxo-N-[3-(phenylsulfanyl)propyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-(4-ethyl-5-methylpyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(6-methoxypyridazin-3-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
6-chloro-N,N-bis(1,3-oxazol-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]thiomorpholine
N5-[(1R)-1-(3-methoxyphenyl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N,N-bis(pyridin-4-ylmethyl)acetamide