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(1R,5R)-6-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(furan-2-ylmethyl)-N-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-oxobutanamide
2,5-dimethyl-3-(4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
(4aR,7aS)-1-cyclopropanecarbonyl-4-(4-methyl-1,3-oxazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 4-({3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}amino)benzoate
2-{2-[1-(1-ethyl-1H-indole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
4-methoxy-2-(4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazin-1-yl)pyrimidine
1-[(5-ethylfuran-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
4-[2-(4-acetylphenoxy)acetyl]-3-(2-hydroxyethyl)piperazin-2-one
1-cyclopentyl-5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-N-methyl-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N3-[2-(4-chlorophenyl)ethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-amino-4-[4-(2-hydroxyethoxy)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-amino-6-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-4-(piperidin-4-yl)pyridine-3-carbonitrile
2-(cyclopropylmethyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
4-chloro-3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H-pyrazole
N-(3-cyclopentylpropyl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methylbenzamide
N5-[1-(furan-2-yl)ethyl]-N3-methyl-4-oxo-N3-(2-phenylethyl)-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
7-chloro-2-methyl-4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
N-(1H-imidazol-2-ylmethyl)-N-methyl-4-(thiophen-2-yl)butanamide
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-4-fluoro-N-(2-methoxyethyl)benzamide
8-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}quinoline
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
2-methyl-6-[3-(morpholine-4-carbonyl)piperidine-1-carbonyl]-4H-pyran-4-one
3-(3-methylbut-2-en-1-yl)-1-(1H-1,2,3-triazole-5-carbonyl)piperidine-3-carboxylic acid
(3S,4S)-1-(3,5-dichloro-4-methylbenzoyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-(morpholin-3-yl)-N-{2-[2-(pyridin-2-yl)ethoxy]phenyl}acetamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-2-(4-propanoylphenoxy)acetamide
N-cyclopropyl-3-[5-(2-methylbutanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
[(3R,5R)-1-(3-ethyl-1,2-oxazole-5-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
1-(4-methoxyphenyl)-3-methyl-4-[3-(morpholin-4-yl)propanoyl]piperazin-2-one
1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(furan-2-yl)propan-1-one
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
3-[ethyl({[2-(furan-2-yl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
9-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]-6-oxa-9-azaspiro[4.5]decane
N-{[(2S,4S)-1-[3-(benzenesulfonyl)propanoyl]-4-fluoropyrrolidin-2-yl]methyl}propanamide
1-(furan-2-ylmethyl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]piperidin-4-amine
4-(1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)benzoic acid
1-[3-(benzyloxy)azetidin-1-yl]-2-(2,4-dichlorophenoxy)ethan-1-one
2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
7-methoxy-3-{[4-methyl-3-oxo-2-(propan-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-{1-[2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]propanamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
N-[4-(1H-pyrazol-5-yl)phenyl]-1-(thian-4-yl)piperidine-3-carboxamide
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide