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5-benzyl-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2S)-1-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidine-2-carboxamide
7-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-(3-{1-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-2-yl}phenoxy)ethan-1-ol
2-[2-(dimethylamino)ethyl]-9-(2,3-dimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3,4-diethoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-[(3-methylphenyl)methyl]piperazine
1-[(3-methylphenyl)methyl]-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
N-(3-benzamido-4-methoxyphenyl)-3-methyl-1H-pyrazole-4-carboxamide
{5-[1-(1-benzothiophen-3-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
5-acetyl-N,2,4-trimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrrole-3-carboxamide
3-hydroxy-1-(2-phenylethyl)-3-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
5-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)morpholine-2-carboxamide
methyl 4-{[cyclohexyl(pyridin-4-ylmethyl)carbamoyl]amino}benzoate
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
3-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)-4H-chromen-4-one
2-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
N,N-dimethyl-3-[2-({[1-(4-methylpyridin-2-yl)propyl]carbamoyl}amino)phenyl]propanamide
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]ethan-1-one
(3aR,6aR)-2-cyclopentyl-5-(cyclopropanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-1-(piperidin-1-yl)propan-1-one
6-(4-hydroxypiperidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)-5-oxopyrrolidine-3-carboxamide
(4aR,7aS)-1-(2-ethylbutanoyl)-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-2-one
4-chloro-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-hydroxy-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N-(2-methoxy-2-methylpropyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
N-(furan-2-ylmethyl)-N,5-dimethyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
1-(morpholin-4-yl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethan-1-one
(1S,5R)-6-(pyridin-2-ylmethyl)-3-[3-(pyridin-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,9aR)-1-[(5-methoxy-1H-1,3-benzodiazol-1-yl)methyl]-octahydro-1H-quinolizin-1-ol
1-(3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}phenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[5-oxo-2-(thiophen-2-yl)cyclopent-1-en-1-yl]acetamide
N-[2-methyl-1-(pyridin-2-yl)propyl]-2-(7-methyl-2-oxo-2H-chromen-4-yl)acetamide
N-[(5-methylthiophen-2-yl)methyl]-6-oxo-N-(prop-2-en-1-yl)-1,6-dihydropyridine-3-carboxamide
2-(2,3-dihydro-1H-inden-5-yloxy)-2-methyl-N-(1,2-oxazol-3-ylmethyl)propanamide
N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}cyclohex-1-ene-1-carboxamide
ethyl 4-(2-phenoxyethyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidine-4-carboxylate
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1,2-oxazole-3-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-cyclobutanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,9R)-11-[3-(2H-1,3-benzodioxol-5-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
(2R,3R)-3-amino-1'-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(4-ethyl-1H-pyrazol-5-yl)-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidine
N-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-1,2,2,6,6-pentamethylpiperidin-4-amine
6-{4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile