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3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(5-fluoropyridin-3-yl)-3-methylurea
(2S,4S)-1-benzyl-N-ethyl-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]pyrrolidine-2-carboxamide
N,2-dimethyl-2-({1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
N-[1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
N-(4,6-dimethylpyridin-2-yl)-3-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)benzamide
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}({[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl})amine
N-[2-(1H-pyrazol-1-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(2E)-3-(2-chlorophenyl)-N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]prop-2-enamide
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
4-{1-[2-(4-hydroxyphenyl)ethyl]-1H-imidazol-2-yl}benzoic acid
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-[4-(5-ethylpyridin-2-yl)-1H-1,2,3-triazol-1-yl]-N-methylethane-1-sulfonamide
2-[1-(furan-2-ylmethyl)-1H-imidazol-2-yl]-1-(propan-2-yl)-1H-1,3-benzodiazole
1-(1-cyclohexylpiperidin-3-yl)-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
ethyl N-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-methylpyrrolidin-3-yl]carbamate
3-(4-methyl-1,3-thiazol-5-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
8-chloro-2-({[2-hydroxy-2-(4-hydroxyphenyl)ethyl]amino}methyl)quinolin-4-ol
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-(4-propylpyrimidine-5-carbonyl)-8-azabicyclo[3.2.1]octane
1-[1-(6-methoxypyrimidin-4-yl)piperidin-3-yl]pyrrolidin-2-one
1-(4-chloro-2-methylphenyl)-3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
3-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
2-(3-methoxypropyl)-9-(quinolin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(4-fluorophenyl)-7-(pyridine-2-amido)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-[4-(difluoromethoxy)phenyl]-3-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
2-({2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)phenol
N-[1-({[3-(1H-indol-1-yl)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]thiophene-3-carboxamide
2-{3-[(4-methylpiperazin-1-yl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl}propanoic acid
2-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-8-fluoroquinoline
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-[(4-hydroxypiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
8-methyl-2-propyl-N-[3-(pyridin-4-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-[(5-propylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
5-{1-[(3-fluorophenyl)methyl]pyrrolidin-2-yl}-N-(2-methoxyethyl)-N-methylthiophene-2-carboxamide
2-(3-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
ethyl 1-(1-{[7-methoxy-2-oxo-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-3-yl]methyl}piperidin-4-yl)piperidine-3-carboxylate
N-cyclopentyl-6-[4-(morpholin-4-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-fluoro-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-phenylethan-1-one
1-ethyl-4-(4-methanesulfonylphenyl)-3-methyl-1H-pyrazole
1-(4-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
5-[1-(3,4-dihydro-2H-1-benzopyran-3-yl)-1H-imidazol-2-yl]-2-(ethylsulfanyl)pyrimidine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[2-(4-fluorophenyl)ethyl]-5-(4-methoxyphenyl)-1,2,4-triazin-3-amine
1-(4-chlorophenyl)-5-methyl-4-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]piperazin-2-one
5-chloro-2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-3-phenyl-1H-indole
N-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-({1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)acetyl]piperidin-4-yl}methyl)benzoic acid