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2-{4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazin-1-yl}pyridine-3-carbonitrile
1-[1'-(2,3-dihydro-1H-indene-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-(3,4-dimethylphenoxy)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
N-({1-[(5-fluoro-2-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)-3-methylbut-2-enamide
8-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(2E)-N-{[4-(cyclooctyloxy)phenyl]methyl}-3-(1H-imidazol-4-yl)-N-(pyridin-3-ylmethyl)prop-2-enamide
3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridazine
(1S,5R)-3-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{1-[(4-chloro-3-fluorophenyl)methyl]pyrrolidin-3-yl}-4-methylpiperazine
N-ethyl-5-[7-fluoro-4-(piperidine-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
2-{1-[3-(piperidin-4-ylmethyl)benzoyl]pyrrolidin-2-yl}pyridine
1-(4-methylpent-3-en-1-yl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-[(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
5-[3-(benzyloxy)propyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
4,6-dimethyl-2-[(1,4-oxazepan-6-ylmethyl)amino]pyridine-3-carbonitrile
N'-(2,4-dimethylphenyl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]ethanediamide
3-(4-hydroxyphenyl)-N-methyl-N-[1-(pyridin-3-yl)pentyl]-1H-pyrazole-5-carboxamide
ethyl 6-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]pyridine-3-carboxylate
1-(azocan-1-yl)-3-{2-methoxy-4-[(4-methoxypiperidin-1-yl)methyl]phenoxy}propan-2-ol
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(3-methylpyridin-2-yl)ethyl]acetamide
methyl 4-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-4-oxobutanoate
2-(dimethyl-1,3-thiazol-5-yl)-N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]acetamide
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{1-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]cyclobutyl}methanol
[(4aS,8aR)-6-[(3,4-dimethoxypyridin-2-yl)methyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(4aS,8aR)-6-[(4-fluoro-3-methoxyphenyl)methyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
(2S,4S)-1-[(2,4-dimethylphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
6-fluoro-2-({[2-methoxy-2-(thiophen-2-yl)ethyl]amino}methyl)quinolin-4-ol
3-[(2-chlorophenyl)methyl]-5-methyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-(furan-2-ylmethyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
methyl 1-(2,4-dimethylpyrimidine-5-carbonyl)piperidine-2-carboxylate
4-(3-fluoropyridin-4-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-(2-chloro-6-methylphenyl)-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholine-4-carboxamide
4-(1H-indol-3-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}butan-1-one
[(3-chloropyridin-4-yl)methyl][2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
N-({1-[(2-aminopyrimidin-5-yl)methyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
5-benzyl-4-[2-(methylamino)acetyl]-1-(3-phenylphenyl)piperazin-2-one
N-(3-ethoxypropyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
(1S,5R)-6-(dimethyl-1,3-oxazole-5-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
ethyl 1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl][(2E)-3-phenylprop-2-en-1-yl]amine
(3R,4S)-3-[(2-aminopyrimidin-4-yl)amino]-N,N-dimethyl-4-(propan-2-yl)pyrrolidine-1-sulfonamide
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-1-methylazepane-2-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[2-(oxan-2-yl)ethyl]propanamide
1-(cyclopropylmethyl)-5-(2-methyloxane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
7-(phenoxathiin-4-yl)-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-[4-(3-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one