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N-methyl-1-(2-phenylethyl)-5-[(prop-2-en-1-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-butyl-1-cyclohexyl-5-[3-(dimethylamino)pyrrolidine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-[3-fluoro-4-(trifluoromethyl)phenyl]-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
3-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-4-(pyridin-3-ylmethyl)piperazin-2-one
N-methyl-2-(2-methyl-1H-1,3-benzodiazol-5-yl)-N-(thiophen-3-ylmethyl)acetamide
N-(2-ethyl-1,3-dihydroxypropan-2-yl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
2-({[2-(dimethylamino)ethyl][(3-methylthiophen-2-yl)methyl]amino}methyl)-6-methylphenol
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-({3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-6-methoxyphenol
N-(3-hydroxypropyl)-N-(naphthalen-1-ylmethyl)-3-(2-oxopiperidin-1-yl)propanamide
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-(3-hydroxyphenyl)pyrrolidin-2-one
4-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}-2,6-dimethoxyphenol
4-(3-chloro-4-hydroxybenzoyl)-1-(4-methylphenyl)piperazin-2-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[3-(pyridin-2-ylmethoxy)phenyl]methyl}amine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)pyrazine-2-carboxamide
5-acetyl-N,2,4-trimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrrole-3-carboxamide
N-[(3R,5S)-1-cycloheptyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
8-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-[1-(2,3-dihydro-1H-inden-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
4-cyclobutaneamido-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]benzamide
3-cyclopropyl-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
N-(2-methyl-2H-1,2,3-triazol-4-yl)-5-{1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-methoxy-4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]quinoline
methyl 6-{[(2-methoxy-2-oxoethyl)(methyl)amino]methyl}-3-(2-phenylacetamido)thieno[2,3-b]pyridine-2-carboxylate
(3R,4S)-4-{ethyl[(2-ethylpyrimidin-4-yl)methyl]amino}oxolan-3-ol
N-[(3R,4R)-1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
1-[9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carbonyl]cyclopropane-1-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]benzamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-N-(propan-2-yl)-2-(thiophen-2-yl)acetamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2,7,8-trimethylquinoline-4-carboxamide
methyl 3-[(pyridin-2-ylformamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
1-ethyl-3-methyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]piperidine-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide
{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(oxan-2-ylmethyl)piperidin-4-yl}methanol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(1-ethyl-1H-pyrazol-3-yl)methyl]-N-methylacetamide
2-(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-2-oxopiperazin-1-yl)benzonitrile
[(4aS,8aR)-6-(2,1,3-benzoxadiazole-4-sulfonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
4-[(2-methylphenyl)sulfanyl]-1-(5-propyl-1,2-oxazole-4-carbonyl)piperidine
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(quinolin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(cyclohex-3-en-1-ylmethyl)amino]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-5-[(propan-2-yl)sulfamoyl]benzamide
2-methoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
1-(2,3-dihydro-1H-indene-5-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-(4-methoxybenzenesulfonyl)-4-(2-methyl-1,3-thiazole-4-carbonyl)piperazine
3,4-difluoro-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
4-methoxy-N-(2-methoxyethyl)-2-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}oxy)benzamide