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2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyridine-3-carbonitrile
[(3R,4R)-1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-(3-fluoro-4-hydroxyphenyl)-1-[3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
(3aR,6aR)-2-cyclohexyl-5-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-ethyl-6-methyl-5-(2-oxo-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
(3aS,7aR)-2-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-{1-[(2-fluorophenyl)methyl]-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
2-{4-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(2-ethylbutyl)-8-[2-(methylamino)-2-phenylacetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)[1-(3-methylpyridin-2-yl)propan-2-yl]amine
N-(3-methylcinnolin-5-yl)-3-(thiophene-2-carbonyl)piperidine-1-carboxamide
2-{4-[(1R,7S)-3-tert-butyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]piperazin-1-yl}acetamide
methyl 3-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}propanoate
2-amino-7-(1H-1,3-benzodiazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2H-1,3-benzodioxole-5-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-methoxyphenyl)-5-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[3-(3-aminoazepan-1-yl)propyl]methanesulfonamide
6-hydroxy-N-(1H-imidazol-2-ylmethyl)-N,2,5,7,8-pentamethyl-3,4-dihydro-2H-1-benzopyran-2-carboxamide
5-methanesulfonyl-N-[(4-methoxyphenyl)methyl]-N-methyl-4-(piperidin-3-yl)pyrimidin-2-amine
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(3-methoxyphenyl)-3-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}propanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(prop-2-en-1-yl)acetamide
2-{2-[(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)methyl]phenoxy}acetic acid
2-amino-3-ethyl-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
1-[3-(2-fluorophenyl)-3-phenylpropanoyl]-1,4-diazepan-5-one
4-(2-fluorophenyl)-2-[5-(methoxymethyl)-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
2-(ethylamino)-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]pyrimidine-5-carboxamide
2-butyl-8-(3-chloro-4-hydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-[3-(pyridin-4-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-benzyl-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2-aminopyrimidin-5-yl)methyl]-1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(4S,6R)-N-[(4-fluorophenyl)methyl]-6-methyl-N-(prop-2-en-1-yl)-2-sulfanylidene-1,3-diazinane-4-carboxamide
3-{[1-(3-cyanopyridin-2-yl)pyrrolidin-3-yl]methyl}benzamide
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-methyl-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
N-butyl-2-[1-(2,4-dimethylpyrimidin-5-yl)-N-methylformamido]acetamide
4-(1-benzofuran-2-yl)-6-methoxypyrimidin-2-amine
(3R,4S)-4-(4-methoxyphenyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-3-amine
N,N-dimethyl-2-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}acetamide
2-butyl-8-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-2-methyl-N-(oxolan-2-ylmethyl)-4-phenylpyridine-3-carboxamide
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
5-(azetidin-1-ylmethyl)-2-(naphthalen-2-yl)pyrimidine
2-(phenylamino)-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidine-5-carboxamide
2-[3-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)phenoxy]pyrimidine
3-(1H-imidazol-2-yl)-6-methoxyquinolin-2-ol
2-methyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)imidazo[1,2-a]pyridine-6-carboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(3-methoxyphenoxymethyl)piperidine