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3-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1H-indole
thiophen-2-yl({1-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]piperidin-4-yl})methanol
1-[3-(dimethylsulfamoyl)-5-{[(2-methylphenyl)methyl]amino}benzoyl]piperidine-3-carboxamide
(3R,4R)-1-(4,5-dimethylthiophene-2-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
[2-(4,6-dimethylpyrimidin-2-yl)ethyl]({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl})amine
1-[(3,5-dimethylphenyl)methyl]-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
4-(2,2-diphenylethyl)-3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]piperazin-2-one
7,7-dimethyl-2-(1-methyl-4-phenylpiperidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
9-(2,6-dimethoxybenzoyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-9-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
4-{[3-(2-aminoethyl)piperidin-1-yl]methyl}-5-chloro-2-methoxyphenol
4-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)pyridine
[(3-ethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
6-hydroxy-7-methoxy-4-[4-(pyrimidin-2-yloxy)phenyl]-1,2,3,4-tetrahydroquinolin-2-one
(1S,5R)-6-(3-fluoropyridine-4-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(2-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)phenyl]imidazolidin-2-one
3-(5-methylthiophen-2-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)-1H-pyrazole-5-carboxamide
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-N,6-dimethyl-4-oxo-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-benzyl-3-[1-(oxan-4-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-7-methoxy-5H,6H-benzo[h]quinoline-3-carbonitrile
2-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-2,7-diazaspiro[4.5]decane
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
N-(1,4-dioxan-2-ylmethyl)-N-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
methyl 2-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)piperidine-1-carboxylate
1-benzyl-5-[(3-methoxyphenyl)methyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]carbamoyl}-1H-imidazole-4-carboxylic acid
2-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
4-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-7-methyl-2H-chromen-2-one
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(1-methyl-1H-indol-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[6-(6-aminopyrimidin-4-yl)-2-(dimethylamino)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
4-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]thiomorpholine
1-[4-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]imidazolidine-2,4-dione
1-[(3,5-dimethylphenyl)methyl]-4-(2-ethylpyridine-4-carbonyl)piperazin-2-one
methyl 1-[(3R,5S)-1-[(4-acetamidophenyl)methyl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-(1-methylpiperidin-3-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]propanamide
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-2-(morpholin-3-yl)acetamide
2-chloro-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}pyridine-4-carboxamide
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-5-(propan-2-yl)pyrimidine
1-{2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}piperidin-2-one
2,5-dimethyl-3-{4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazin-1-yl}pyrazine
7-acetamido-2-(2-methoxyphenyl)-1-methyl-N-[3-(pyridin-3-yloxy)propyl]-1H-1,3-benzodiazole-5-carboxamide
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-1-methyl-1H-1,3-benzodiazole
6-fluoro-N-methyl-2-oxo-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl (2S)-3-(1H-imidazol-4-yl)-2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propanoate
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(pyrrolidin-1-yl)propan-1-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1H-1,2,3-benzotriazole-5-carboxamide
1-(1-ethyl-1H-pyrazole-3-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
6-{[benzyl(ethyl)amino]methyl}-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide