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2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}acetamide
5-[({[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
(isoquinolin-5-ylmethyl)(methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-1-methyl-1H-indole
(3S)-3-ethyl-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}morpholine
3-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-phenylpropanamide
1-(2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1-methylurea
4-methyl-2-(propan-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1,3-thiazole-5-carboxamide
2-methyl-N-(thiolan-3-yl)imidazo[1,2-a]pyridine-6-carboxamide
(oxolan-2-ylmethyl)({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(thiophen-3-ylmethyl)amine
(3S,4S)-1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-fluoro-N-methyl-5-({[1-(oxan-4-yl)piperidin-4-yl]carbamoyl}amino)benzamide
ethyl(methyl){[(3R,4S)-4-(propan-2-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-3-yl]sulfamoyl}amine
N-methyl-N-({1-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)furan-2-carboxamide
3-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1-propyl-1H-pyrazole-4-carboxamide
1-[4-methyl-2-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)pyrimidin-5-yl]ethan-1-one
N-{[4-(hydroxymethyl)phenyl]methyl}-2,6-dimethylpyridine-4-carboxamide
3-(2-phenylethyl)-1-(quinoxalin-2-yl)piperidine-3-carboxylic acid
2-methyl-7-[(4-methyl-2-oxo-2H-chromen-7-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-{4-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-N'-cycloheptylbutanediamide
1-[2-(4-methoxyphenyl)ethyl]-N-[2-(methylsulfanyl)ethyl]-6-oxopiperidine-3-carboxamide
8-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{ethyl[(4-ethylphenyl)methyl]amino}propane-1,2-diol
1-(1-ethylpiperidin-3-yl)-4-(piperidin-1-yl)piperidine
4-{[3-(1-benzyl-1H-pyrazol-4-yl)phenyl]methyl}morpholine
N-(1-benzothiophen-5-ylmethyl)-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
6-fluoro-3-[2-(4-hydroxypiperidin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
4-({2-[1-(ethanesulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[3-(benzyloxy)propyl]-1,3-diazinane-2,4-dione
N-[4-(6-methyl-9H-purin-9-yl)phenyl]acetamide
N-[(3S)-2-oxoazepan-3-yl]imidazo[1,2-a]pyridine-6-carboxamide
5-(2-methoxyacetamido)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
6-[4-(5-methoxy-1-methyl-1H-indole-2-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
methyl 7-oxo-9-(pyridin-2-ylmethoxy)-3-[2-(1,3-thiazol-4-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(3,3-diphenylpiperidin-1-yl)-2-(pyrrolidin-1-yl)ethane-1,2-dione
N-methyl-N-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
7-[(4-fluorophenyl)methyl]-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,9aR)-8-(4-ethylbenzoyl)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(4-chloro-2-methoxyphenoxymethyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
N-(pyridin-3-ylmethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
(but-2-yn-1-yl)(furan-2-ylmethyl){[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
N-benzyl-N-methyl-3-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]propanamide
3-(1H-imidazol-2-yl)-2-methoxyquinoline
4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}butanamide
4-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1H-imidazole-5-carboxamide
N,N-dimethyl-3-[(2-methyl-5-propylpyrimidin-4-yl)amino]azepane-1-sulfonamide
N'-benzyl-N'-(3-hydroxy-2-methylpropyl)-N,N-dimethylbutanediamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(quinoxalin-2-yl)piperidin-3-yl]propanoic acid