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N-(3-methylphenyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-indazol-3-yl)acetamide
(3aR,6aS)-5-{[4-(2-hydroxyethoxy)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
6-{[(3S,4R)-3-cyclopropyl-4-[(dimethylsulfamoyl)amino]pyrrolidin-1-yl]methyl}-2-methylpyrimidin-4-ol
ethyl 3-({5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazol-4-yl}formamido)propanoate
1-(4-methoxyphenyl)-2,2-dimethyl-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperazine
1-benzyl-8-(furan-2-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(5-acetamido-2-methoxyphenyl)-4-(3-methoxypropyl)piperazine-1-carboxamide
[5-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)furan-2-yl]methanol
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-5-methyl-4,5,6,7-tetrahydro-2H-indazole
4-(5-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
2-amino-4-[3-(2-hydroxyethoxy)phenyl]-5-methyl-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
3-(2H-1,3-benzodioxol-5-yl)-5-(thian-4-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-(3-chloro-4-hydroxyphenyl)ethan-1-one
N,1,7-trimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-indole-2-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidine-3-carboxylate
ethyl 1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[4-({methyl[(3-methylthiophen-2-yl)methyl]carbamoyl}methoxy)phenyl]propanamide
3-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-[3-(hydroxymethyl)-2-methylphenyl]benzamide
3-[4-(hydroxymethyl)phenyl]-4H-chromen-4-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
N-(2-methoxy-5-{[methyl(1-methylpiperidin-4-yl)carbamoyl]amino}phenyl)propanamide
N,N-dimethyl-3-{[1-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)propan-2-yl]oxy}aniline
(2R,3R,6R)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-fluoro-3-[2-(pyridin-3-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
5-{2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-4-(3-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carboxamide
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(pyridin-4-yl)piperazin-1-yl]acetic acid
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
4-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)piperazine-2-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
4-amino-2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidine-5-carbonitrile
4-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}morpholine
3-[({[1-(methoxymethyl)cyclopropyl]methyl}carbamoyl)methyl]-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-methoxypyridine-3-carbonitrile
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-fluoro-5-sulfamoylbenzamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-methyl-1H-imidazole-5-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-3-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-4-cyclopropyl-4-methylpyrrolidin-2-one
1-{2-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]pyrimidin-4-yl}piperidin-3-ol
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-butyl-2-(1H-imidazol-4-yl)-N-(thiophen-3-ylmethyl)acetamide
2-methyl-N-{1-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-(azepan-1-yl)-3-(4-chloro-2-{[(1-methylpiperidin-4-yl)amino]methyl}phenoxy)propan-2-ol
N-[2-(methylsulfanyl)ethyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-cyclopropyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide