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8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
1-cycloheptyl-N-[(5-methylfuran-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
6-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
4-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}pyridine
4-{1-[(2-butyl-1H-imidazol-4-yl)methyl]azetidin-3-yl}pyridine
3-{2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-4-(2-phenylethyl)piperazin-2-one
1-phenyl-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-(2,4-dichlorophenoxy)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]acetamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(3-ethyl-1,2-oxazol-5-yl)methyl]amine
4-[5-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
(3S,4R)-1-(3-carboxybenzoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
13-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
2-{[2-(3-chlorophenyl)-1H-imidazol-1-yl]methyl}-4,6-dimethylpyrimidine
N-{1-azabicyclo[2.2.2]octan-3-yl}-1-(methoxymethyl)cyclobutane-1-carboxamide
1-(4-fluorophenyl)-2-(furan-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-({3-[(dimethylamino)methyl]phenyl}formamido)-N-hydroxybutanamide
2-acetyl-8-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(dimethylamino)-8-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-(pyridin-3-ylmethyl)-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
4-[4-(thiomorpholine-4-carbonyl)benzenesulfonyl]morpholine
5-methyl-4-[(oxolan-3-yl)amino]-N-[2-(4-phenylpiperidin-1-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
1-[4-(3-fluorophenyl)phenyl]-3-methyl-3-[(1-methyl-5-oxopyrrolidin-3-yl)methyl]urea
ethyl 4-(2-phenoxyethyl)-1-(thiolan-3-yl)piperidine-4-carboxylate
7-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N,N-dimethyl-7-(1H-pyrazole-3-carbonyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
4-chloro-N-[2-(1H-imidazol-1-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-(2-hydroxyphenyl)ethan-1-one
methyl[1-(pyridin-3-yl)propyl]{[6-(trifluoromethyl)pyridin-3-yl]methyl}amine
1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-amine
2-(1-ethyl-1H-pyrazol-4-yl)-7-methoxy-N-(oxan-3-yl)quinoline-4-carboxamide
3-{[({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)carbamoyl]amino}-N-(propan-2-yl)benzamide
(1R,5R)-6-(cyclopropylmethyl)-3-(2,6-difluoro-3-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[methyl({[3-(2-{4-[4-(trifluoromethyl)benzenesulfonyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
5-[(4-ethylpiperazin-1-yl)methyl]-N-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-1,2-oxazole-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
(2R,3R,6R)-5-(2-methoxypyridine-3-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-({[2-(2-hydroxyethoxy)ethyl]amino}methyl)-5,8-dimethylquinolin-4-ol
3-(furan-2-yl)-4-pentyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-sulfonyl]-N-(2,2,2-trifluoroethyl)benzamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
ethyl 4-[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]piperidine-1-carboxylate