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N-methyl-3-(2-phenylethyl)-N-(thiophen-3-ylmethyl)-1,2-oxazole-5-carboxamide
4-{3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propoxy}benzamide
4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
(2S,4S)-N-ethyl-1-(oxan-4-yl)-4-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetamido]pyrrolidine-2-carboxamide
2-[methyl(pyridin-3-ylmethyl)amino]-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
N-cyclohexyl-5,7-dimethyl-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[({1-oxaspiro[4.5]decan-3-yl}carbamoyl)amino]benzamide
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methylthiophene-3-carbonyl)piperidine
N-[4-(1H-imidazol-1-yl)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-(4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)acetamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(4-propylpyrimidine-5-carbonyl)pyrrolidin-3-ol
N-phenyl-5-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{[1-(2-aminopyrimidin-4-yl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
N-[(5-{[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
N-methyl-N-[1-(naphthalen-2-yl)ethyl]-3-(pyrazin-2-yl)propanamide
N-[(2,3-difluoro-4-methylphenyl)methyl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
(3R,4S)-3-amino-N-ethyl-N-methyl-4-propylpyrrolidine-1-sulfonamide
N-cyclopropyl-N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-2-phenylethyl]pyridine-2-carboxamide
4-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-methyl-1H-imidazole
N'-(3-chloro-4-methylphenyl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}propanediamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-4-fluorobenzamide
2-(1H-imidazol-1-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-[4-(pyridin-2-yl)pyrimidin-2-yl]pyrrolidin-3-ol
2-{[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
(3R,4R)-1-(1-cyclopentylpiperidine-4-carbonyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
3-{1-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}pyridine
4-{[4-(3-phenylpropyl)-1,4-diazepan-1-yl]methyl}phenol
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(4-methylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
6-chloro-3-fluoro-N-[3-(2-oxopyrrolidin-1-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]urea
methyl[(5-methylfuran-2-yl)methyl]{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}amine
8-[(5-ethylthiophen-2-yl)sulfonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-(3-chlorophenyl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
5-(2-methylpropyl)-1'-(2-methylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[2-methoxy-4-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
N-ethyl-2-[3-(2-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyridine-3-carboxamide
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
1,4-dimethyl-9-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecane
2,8-dimethyl-4-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]quinoline
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(oxan-2-ylmethyl)propanamide
1-cyclopentyl-4-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)piperazine
4-[5-(2,4-dimethylpyrimidin-5-yl)-1,2,4-oxadiazol-3-yl]-1H-indole
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-[2-(dimethylamino)ethyl]-N-[(2-ethoxypyridin-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide