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(3aR,7aS)-N-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
5-ethyl-N-[(3,4,5-trifluorophenyl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-benzylpiperazine-1-carbonyl)-6-[1-(4-chlorophenyl)cyclopropanecarbonyl]-6-azaspiro[2.5]octane
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(1-methyl-1H-indol-5-yl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
1-tert-butyl-4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrrolidin-2-one
1-[4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(pyrrolidin-1-yl)propan-1-one
1-cyclopentyl-4-(2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazin-2-one
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]acetamide
N-[2-(2-chlorophenyl)-1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
7-(3-fluoropyridin-4-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
[(3S,3aS,6aR)-3-(1-ethyl-1H-pyrazol-4-yl)-1-(hydroxymethyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
3-benzyl-4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperazin-2-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
5-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-(4-methoxyphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-(3-methoxyphenyl)-3-{1-[3-(morpholin-4-yl)propanoyl]piperidin-4-yl}propanamide
4-(4-chloro-2-methoxybenzoyl)-1-(4-methoxyphenyl)piperazin-2-one
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-(3-methylcinnolin-5-yl)urea
8-(5-amino-1H-pyrazole-3-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(thiophene-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(2-hydroxyethyl)-2,3-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-indole-5-carboxamide
1-(4-fluoro-2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-one
2-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]isoquinoline
4-cyclopentyl-2-[(3-methoxyphenyl)methyl]morpholine
(2S,4S)-4-amino-N-methyl-1-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}pyrrolidine-2-carboxamide
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-N,N-dimethyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-sulfonamide
1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(propan-2-yl)-1,4-diazepane
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-carboxamide
3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]-N-(2-phenylethyl)piperidine-1-carboxamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
3-(4-fluorophenoxymethyl)-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)piperidine-1-carboxamide
2-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}benzoic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(2,4,6-trimethylphenyl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[1-(3-hydroxyadamantan-1-yl)ethyl]-5-(methoxymethyl)furan-2-carboxamide
3-(2-hydroxyphenyl)-N-{2-[methyl(2-phenylethyl)amino]ethyl}-1H-pyrazole-5-carboxamide
3-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylpropanamide
N-(4-acetylphenyl)-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2,3-dihydro-1,4-benzodioxine-6-carboxamide
3-(1,3-benzothiazol-2-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]propan-1-one
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
8-(2,3-dimethyl-1H-indole-7-carbonyl)-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
7-chloro-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3,5-dimethyl-1-benzofuran-2-carboxamide
4-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-N-(2-phenylethyl)pyridine-2-carboxamide
2-chloro-5-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-1,2,3-triazol-4-yl)pyridine
N-[(3R,4S)-1-(4-aminopyrimidin-2-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
4-[(2,6-dichloro-3-hydroxyphenyl)methyl]piperazine-1-sulfonamide