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5-(2-methoxy-6-methylphenyl)-3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
methyl 8-[(6-chloro-4-oxo-4H-chromen-3-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(2-methyl-4-{methyl[3-(pyrrolidin-1-yl)propyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
1-(2-methoxyphenyl)-4-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine
3-[3-({[(2-fluorophenyl)methyl](2-hydroxyethyl)amino}methyl)-1H-indol-1-yl]propanamide
1-(1-benzothiophen-2-ylmethyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
methyl 4-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}benzoate
3-{2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1λ6-thiolane-1,1-dione
N-benzyl-1-(cyclopropylmethyl)-N-methylpiperidin-3-amine
N-ethyl-1-(furan-2-ylmethyl)-N-(oxan-4-ylmethyl)piperidine-3-carboxamide
2-[4-(4-methyl-1H-pyrrole-2-carbonyl)morpholin-3-yl]-N-[2-(2-methylphenyl)ethyl]acetamide
5-(methoxymethyl)-N-[2-(morpholin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-chlorophenyl)-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)cyclobutane-1-carboxamide
1-(3-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}phenyl)imidazolidin-2-one
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(1,2-oxazol-5-yl)phenol
2-cyclohexyl-6-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
7-[(3,4-difluorophenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decane
3-[(3R,4S)-4-(morpholin-4-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]propan-1-ol
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(4-phenylbenzoyl)piperidine
methyl 8-(1-benzothiophen-2-ylmethyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2,6-dimethylquinoline
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethylacetamide
3-[(3-fluorophenyl)methyl]-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
4-methyl-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,4-diazepan-5-one
4-[3-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)propyl]piperazin-2-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
2-[1-({1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-ol
3-(1-methyl-1H-pyrazol-4-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-amino-6-(2,5-dimethylfuran-3-yl)-4-(4-hydroxyphenyl)pyridine-3-carbonitrile
(2S,4R)-4-amino-N-methyl-1-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)pyrrolidine-2-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-(2-methoxypyrimidine-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-{[(pyridin-2-ylmethyl)carbamoyl]methyl}-1,4-diazepane-6-carboxylic acid
5-methyl-4-(oxane-4-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
N,3,5-trimethyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1-benzofuran-2-carboxamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidine-3-carboxamide
1-(3-phenyl-1H-pyrazole-4-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-[2-(ethylamino)pyrimidine-5-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-ethyl-N-[2-(piperidin-1-yl)ethyl]pyrazolo[1,5-a]pyridine-3-carboxamide
3-{[2-(hydroxymethyl)-1H-1,3-benzodiazol-5-yl]formamido}-N-phenylpropanamide
1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-2-phenylethane-1,2-dione
4-{[7-(cyclohex-1-en-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(3,5-dimethoxybenzoyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
3-[(4-methylphenyl)methyl]-1-{1-[3-(methylsulfanyl)propanoyl]azepan-3-yl}urea
(1S,2S)-N2-(trimethylpyrimidin-4-yl)-2,3-dihydro-1H-indene-1,2-diamine
1-[3-(3-fluorophenyl)phenyl]-3-{3-[3-(hydroxymethyl)piperidin-1-yl]propyl}urea
2-(5-acetylthiophen-3-yl)-1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}ethan-1-one
5-methoxy-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-indole-2-carboxamide
1-(4-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]sulfonyl}phenyl)ethan-1-one
benzyl (7S,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate